SCHEMBL8158593

SCHEMBL8158593

C=CC[N][13c]1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.39
TSHR P16473 2/20 0.36
RAB9A P51151 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
CYP2C19 P33261 3/20 0.33
CYP1A2 P05177 1/20 0.33
GAA P10253 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
ADRA1D P25100 1/20 0.32
ADRA1A P35348 1/20 0.32
ADRA1B P35368 1/20 0.32
MIF P14174 1/20 0.32
HTR3E A5X5Y0 1/20 0.32
SLC22A2 O15244 1/20 0.32
SLC22A1 O15245 1/20 0.32
SLC22A3 O75751 1/20 0.32
HTR3B O95264 1/20 0.32
PLAU P00749 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL44664 1.00 ALDH1A1 (0.39) ALDH1A1TSHRRAB9ASMN1; SMN2CYP2C19
SCHEMBL11767820 0.82 ALDH1A1 (0.50) ALDH1A1TSHRCYP2C19CYP1A2GAA
SCHEMBL7718086 0.76 ALDH1A1 (0.48) ALDH1A1TSHRRAB9ACYP2C19CYP1A2
SCHEMBL10432560 0.76
SCHEMBL3478608 0.76 CYP3A4 (0.40) ALDH1A1TSHRCYP1A2CYP2C9SLC22A2
SCHEMBL7718084 0.76 ALDH1A1 (0.48) ALDH1A1TSHRRAB9ACYP2C19CYP1A2
SCHEMBL8517746 0.75 ALDH1A1 (0.39) ALDH1A1RAB9ACYP2D6MIFHTR3E
SCHEMBL8083518 0.72 MIF (0.40) ALDH1A1TSHRRAB9ACYP2C19CYP1A2
SCHEMBL10443511 0.70 ALDH1A1 (0.35) ALDH1A1MIF
SCHEMBL7775723 0.70 ALDH1A1 (0.41) ALDH1A1TSHRSMN1; SMN2CYP2C19CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0871619-A1 PHENYL THIAZOLE DERIVATIVES WITH ANTI HERPES VIRUS PROPERTIES BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 1998-10-21 EP claimed
WO-1997024343-A1 PHENYL THIAZOLE DERIVATIVES WITH ANTI HERPES VIRUS PROPERTIES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 1997-07-10 WO claimed
EP-0315367-B1 Polypeptides ICI PLC (GB) 1994-04-06 EP claimed
US-5081107-A Bombesin or bombesin-like peptides antagonists; anticarcinogenic agents; antisecretory agents; glandular disorders IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-01-14 US claimed
US-5068222-A Polypeptides for treatment of cancer IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-11-26 US claimed
EP-0345990-A2 Polypeptide compounds ZENECA LIMITED (GB) 1989-12-13 EP claimed
EP-0315367-A2 Polypeptides IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1989-05-10 EP claimed
JP-1151599-A None JP disclosed
US-6057451-A AMINOTHIAZOLE DERIVATIVES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2000-05-02 US disclosed
EP-0871619-A1 PHENYL THIAZOLE DERIVATIVES WITH ANTI HERPES VIRUS PROPERTIES BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 1998-10-21 EP disclosed
WO-1997024343-A1 PHENYL THIAZOLE DERIVATIVES WITH ANTI HERPES VIRUS PROPERTIES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 1997-07-10 WO disclosed
EP-0315367-B1 Polypeptides ICI PLC (GB) 1994-04-06 EP disclosed
US-5081107-A Bombesin or bombesin-like peptides antagonists; anticarcinogenic agents; antisecretory agents; glandular disorders IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-01-14 US disclosed
US-5068222-A Polypeptides for treatment of cancer IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-11-26 US disclosed
EP-0345990-A2 Polypeptide compounds ZENECA LIMITED (GB) 1989-12-13 EP disclosed
JP-H01151599-A POLYPEPTIDE, ITS PREPARATION AND PHARMACEUTICAL COMPOSITION USED IN TREATMENT OF DISEASES OR MEDICAL CONDITION ARRANGED BY BOMBESIN OR BOMBESIN-LIKE PEPTIDE IMPERIAL CHEM IND PLC <ICI> 1989-06-14 JP disclosed
EP-0315367-A2 Polypeptides IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1989-05-10 EP disclosed