SCHEMBL8159362

SCHEMBL8159362

O=S(=O)(c1c(Cl)ccc2nonc12)N1CCC(Oc2ncccn2)CC1

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.58
NPC1 O15118 1/20 0.58
TLR9 Q9NR96 1/20 0.58
ALDH1A1 P00352 4/20 0.42
NAAA Q02083 1/20 0.41
MEN1 O00255 3/20 0.39
POLB P06746 1/20 0.39
FPR2 P25090 7/20 0.39
PROKR1 Q8TCW9 7/20 0.39
MAPT P10636 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
EPHX2 P34913 1/20 0.38
CYP2J2 P51589 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6390286 0.88 KMT2A (0.45) KMT2ANPC1TLR9ALDH1A1NAAA
SCHEMBL5243713 0.85 ALDH1A1 (0.43) KMT2ANPC1TLR9ALDH1A1NAAA
SCHEMBL5243164 0.83 ALDH1A1 (0.60) KMT2AALDH1A1MEN1POLBCYP2C19
SCHEMBL5244612 0.80 NPC1 (0.53) KMT2ANPC1TLR9FPR2PROKR1
SCHEMBL5285381 0.72 KMT2A (0.58) KMT2ANPC1TLR9ALDH1A1MEN1
SCHEMBL5288051 0.71 KMT2A (0.57) KMT2ANPC1TLR9ALDH1A1MEN1
SCHEMBL5281618 0.71 KMT2A (0.49) KMT2ANPC1TLR9ALDH1A1MEN1
SCHEMBL5244644 0.71 KMT2A (0.62) KMT2ANPC1TLR9ALDH1A1MEN1
SCHEMBL5244144 0.69 ALDH1A1 (0.40) KMT2AALDH1A1MEN1POLBMAPT
SCHEMBL5290061 0.69 SCD (0.47) FPR2PROKR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008115259-A2 DERIVATIVES OF BENZOXADIAZOLE SUITABLE FOR THE TREATMENT OF CELL PROLIFERATIVE DISEASES RIGEL PHARMACEUTICALS, INC. (US) 2008-09-25 WO disclosed
WO-2006002284-A1 UBIQUITIN LIGASE INHIBITORS RIGEL PHARMACEUTICALS, INC. (US) 2006-01-05 WO disclosed