SCHEMBL8164149

SCHEMBL8164149

CCc1cc(Br)ccc1CC(=O)N1C(=O)OC[C@H]1Cc1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NAAA Q02083 3/20 0.40
PPARA Q07869 4/20 0.39
BRD4 O60885 1/20 0.37
PPARG P37231 1/20 0.36
ALDH1A1 P00352 2/20 0.36
IL6ST P40189 1/20 0.36
KDM4E B2RXH2 1/20 0.36
FAAH O00519 1/20 0.36
CSNK2B P67870 1/20 0.36
CSNK2A1 P68400 1/20 0.36
HDAC1 Q13547 2/20 0.35
IDH1 O75874 3/20 0.35
CCR3 P51677 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3308822 0.90 NAAA (0.41) NAAAPPARABRD4PPARGIL6ST
SCHEMBL3308816 0.90 NAAA (0.41) NAAAPPARABRD4PPARGIL6ST
SCHEMBL16737997 0.90 NAAA (0.41) NAAAPPARABRD4PPARGIL6ST
SCHEMBL24977629 0.88 NAAA (0.45) NAAAPPARAPPARGALDH1A1IL6ST
SCHEMBL2553570 0.88 AKR1B1 (0.39) NAAAPPARA
SCHEMBL8164388 0.88 NAAA (0.38) NAAAPPARABRD4ALDH1A1IL6ST
SCHEMBL2552573 0.88 AKR1B1 (0.39) NAAAPPARA
SCHEMBL15092485 0.88 AKR1B1 (0.39) NAAAPPARA
SCHEMBL3305644 0.87 KDM4E (0.45) NAAAALDH1A1KDM4ECSNK2BCSNK2A1
SCHEMBL3305638 0.87 KDM4E (0.45) NAAAALDH1A1KDM4ECSNK2BCSNK2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008079836-A2 MACROCYCLIC FACTOR VIIA INHIBITORS USEFUL AS ANTICOAGULANTS BRISTOL-MYERS SQUIBB COMPANY (US) 2008-07-03 WO disclosed