SCHEMBL8166156

SCHEMBL8166156

CCCCn1ccc(-c2ccc(Oc3cc(C)nc(C)c3)c(F)c2)c(N)c1=O

nearest known ligand 0.75

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 20/20 0.75

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2831204 0.86 GRM2 (1.00) GRM2
SCHEMBL8152779 0.82 GRM2 (0.62) GRM2
SCHEMBL2830396 0.77 GRM2 (1.00) GRM2
SCHEMBL2829844 0.74 GRM2 (0.81) GRM2
SCHEMBL2831836 0.71 GRM2 (0.83) GRM2
SCHEMBL2186805 0.71 GRM2 (0.65) GRM2
SCHEMBL30795860 0.71 GRM2 (0.65) GRM2
SCHEMBL2831898 0.70 GRM2 (0.73) GRM2
SCHEMBL8167358 0.68 GRM2 (0.51) GRM2
SCHEMBL8157229 0.66 GRM2 (0.49) GRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008107480-A1 1,4-DISUBSTITUTED 3-CYANO-PYRIDONE DERIVATIVES AND THEIR USE AS POSITIVE MGLUR2 -RECEPTOR MODULATORS ORTHO-MCNEIL-JANSSEN PHARMACEUTICALS, INC (US) 2008-09-12 WO disclosed