SCHEMBL8167387

SCHEMBL8167387

Cn1nc(-c2ccc(S(C)(=O)=O)cc2)c(-c2ccc(Cl)cc2)c1C(=O)O

nearest known ligand 0.46

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 4/20 0.46
PTGS2 P35354 10/20 0.46
CA12 O43570 1/20 0.45
CA9 Q16790 1/20 0.45
FAAH O00519 2/20 0.43
KCNH2 Q12809 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8179845 0.89 PTGS2 (0.55) PTGS1PTGS2CA12CA9
SCHEMBL8179842 0.89 PTGS2 (0.53) PTGS1PTGS2CA12CA9
SCHEMBL7773091 0.88 PTGS2 (0.46) PTGS1PTGS2CA12CA9
SCHEMBL7777656 0.88 PTGS2 (0.46) PTGS1PTGS2CA12CA9
SCHEMBL7777967 0.84 PTGS2 (0.52) PTGS1PTGS2CA12CA9
SCHEMBL8975526 0.84 PTGS1 (0.43) PTGS1PTGS2CA12CA9
SCHEMBL8180056 0.84 PTGS2 (0.45) PTGS1PTGS2CA12CA9FAAH
SCHEMBL8634798 0.82 PTGS1 (0.42) PTGS1PTGS2CA12CA9FAAH
SCHEMBL7778046 0.82 PTGS2 (0.52) PTGS1PTGS2FAAHKCNH2
SCHEMBL7773163 0.81 PTGS2 (0.58) PTGS1PTGS2CA12CA9FAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6028072-A 3,4-substituted pyrazoles for the treatment of inflammation G. D. SEARLE & CO. (US) 2000-02-22 US disclosed
US-5486534-A 3,4-substituted pyrazoles for the treatment of inflammation G. D. SEARLE & CO. (US) 1996-01-23 US disclosed