SCHEMBL81677

SCHEMBL81677

Cc1ccc(-c2ccc3c(c2)C(C)(C)c2cc(-c4ccc5c(c4)-c4cccnc4C5(C)C)ccc2-3)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 10/20 0.42
COMT P21964 1/20 0.35
PGR P06401 1/20 0.34
AKT1 P31749 1/20 0.32
BACE1 P56817 1/20 0.32
KCNH2 Q12809 1/20 0.32
GRM5 P41594 1/20 0.32
SYK P43405 1/20 0.32
FLT3 P36888 1/20 0.31
TNKS2 Q9H2K2 1/20 0.31
NPC1 O15118 1/20 0.31
ALDH1A1 P00352 1/20 0.31
CYP1A2 P05177 1/20 0.31
GAA P10253 1/20 0.31
MAPT P10636 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
RAB9A P51151 1/20 0.31
MCL1 Q07820 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL92299 0.88 PDK2 (0.44) PDK2SYKNPC1ALDH1A1RAB9A
SCHEMBL22373946 0.81 PDK2 (0.46) PDK2COMTTNKS2NPC1ALDH1A1
SCHEMBL22373903 0.81 PDK2 (0.41) PDK2TNKS2NPC1ALDH1A1CYP1A2
SCHEMBL81678 0.81 PDK2 (0.40) PDK2NPC1ALDH1A1MAPTRAB9A
SCHEMBL81604 0.77 PDK2 (0.41) PDK2CYP1A2GAACYP2C19
SCHEMBL81614 0.77 PDK2 (0.41) PDK2CYP1A2GAACYP2C19
SCHEMBL19928405 0.76 PDK2 (0.44) PDK2
SCHEMBL81615 0.76 PDK2 (0.39) PDK2PGRBACE1NPC1CYP1A2
SCHEMBL24810030 0.75 L3MBTL1 (0.40) PDK2FLT3NPC1ALDH1A1GAA
SCHEMBL9963989 0.75 PDK2 (0.41) PDK2PGRKCNH2NPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129899-B1 Azafluorene derivative and organic light-emitting device using the derivative CANON KABUSHIKI KAISHA (JP) 2012-03-06 US disclosed
US-20120049176-A1 AZAFLUORENE DERIVATIVE AND ORGANIC LIGHT-EMITTING DEVICE USING THE DERIVATIVE CANON KABUSHIKI KAISHA (JP) 2012-03-01 US disclosed