SCHEMBL8168274

SCHEMBL8168274

Cc1cc(C)c(S(=O)(=O)N[C@@H](CNC(=O)c2nnc(CCCCNc3ccccn3)s2)C(=O)O)c(C)c1

nearest known ligand 0.63

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 14/20 0.63
ITGAV P06756 14/20 0.63
ITGA2B P08514 9/20 0.63
ITGB1 P05556 8/20 0.50
ITGA5 P08648 8/20 0.50
ITGB5 P18084 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8168263 1.00 ITGB3 (0.63) ITGB3ITGAVITGA2BITGB1ITGA5
SCHEMBL7369516 0.84 ITGB3 (0.48) ITGB3ITGAVITGA2BITGB1ITGA5
SCHEMBL8179651 0.83 ITGAV (0.63) ITGB3ITGAVITGA2BITGB1ITGA5
SCHEMBL8179647 0.83 ITGAV (0.63) ITGB3ITGAVITGA2BITGB1ITGA5
SCHEMBL8176082 0.83 ITGAV (0.65) ITGB3ITGAVITGA2BITGB1ITGA5
SCHEMBL6495549 0.82 ITGAV (0.63) ITGB3ITGAVITGA2BITGB1ITGA5
Acetic Acid SCHEMBL6504819 0.80 ITGAV (0.61) ITGB3ITGAVITGA2BITGB1ITGA5
SCHEMBL8176077 0.78 ITGAV (0.46) ITGB3ITGAVITGA2BITGB1ITGA5
SCHEMBL7403221 0.78 ITGB3 (1.00) ITGB3ITGAVITGA2B
SCHEMBL7369530 0.78 ITGB3 (0.41) ITGB3ITGAVITGA2BITGB1ITGA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153628-A 1,3,4-thiadiazoles and 1,3,4-Oxadiazoles as αv β3 antagonists DUPONT PHARMACEUTICALS COMPANY (US) 2000-11-28 US claimed
US-6153628-A 1,3,4-thiadiazoles and 1,3,4-Oxadiazoles as αv β3 antagonists DUPONT PHARMACEUTICALS COMPANY (US) 2000-11-28 US disclosed