SCHEMBL8169010

SCHEMBL8169010

Cc1cc(-c2ccc(C=O)cc2)cc(-n2c(=O)n(C3CCC(NC(=O)c4cn5cc(F)ccc5n4)CC3)c(=O)c3cc(F)cnc32)c1

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 8/20 0.43
CNR2 P34972 5/20 0.36
CNR1 P21554 4/20 0.35
HPGDS O60760 2/20 0.35
GPR55 Q9Y2T6 1/20 0.35
ABL1 P00519 2/20 0.34
DPP4 P27487 1/20 0.33
USP30 Q70CQ3 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL870691 1.00 PDE4B (0.43) PDE4BCNR2CNR1HPGDSGPR55
SCHEMBL870690 1.00 PDE4B (0.43) PDE4BCNR2CNR1HPGDSGPR55
SCHEMBL870026 0.92 PDE4B (0.45) PDE4BCNR2CNR1HPGDS
SCHEMBL870027 0.92 PDE4B (0.45) PDE4BCNR2CNR1HPGDS
SCHEMBL870639 0.91 PDE4B (0.45) PDE4BCNR2CNR1
SCHEMBL870249 0.89 PDE4B (0.42) PDE4BCNR2CNR1HPGDSGPR55
SCHEMBL870250 0.89 PDE4B (0.42) PDE4BCNR2CNR1HPGDSGPR55
SCHEMBL8170582 0.87 PDE4B (0.46) PDE4BCNR2CNR1HPGDSGPR55
SCHEMBL870978 0.87 PDE4B (0.46) PDE4BCNR2CNR1HPGDSGPR55
SCHEMBL870977 0.87 PDE4B (0.46) PDE4BCNR2CNR1HPGDSGPR55

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008084223-A2 CHEMICAL COMPOUNDS 637: PYRIDOPYRIMIDINEDIONES AS PDE4 INHIBITORS ASTRAZENECA AB (SE) 2008-07-17 WO disclosed