SCHEMBL8169472

SCHEMBL8169472

COC(=O)c1ccc(-c2nc(NCc3ccc(OC)c(Cl)c3)c3c(C)csc3n2)cc1

nearest known ligand 0.47

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.47
BCDIN3D Q7Z5W3 2/20 0.41
PDE5A O76074 8/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8171015 0.93 ESR1 (0.47) ESR1BCDIN3DPDE5AMEN1KMT2A
SCHEMBL8184899 0.92 ESR1 (0.49) ESR1MEN1KMT2A
SCHEMBL8179394 0.92 MEN1 (0.48) ESR1MEN1KMT2A
SCHEMBL5115035 0.88 ESR1 (0.48) ESR1BCDIN3DPDE5AMEN1KMT2A
SCHEMBL8182349 0.86 PRKCI (0.43) BCDIN3DPDE5AKMT2A
SCHEMBL8177950 0.86 BCDIN3D (0.41) BCDIN3DPDE5AMEN1KMT2A
SCHEMBL5814645 0.85 ESR1 (0.46) ESR1BCDIN3DPDE5AMEN1KMT2A
SCHEMBL8171050 0.85 KMT2A (0.50) ESR1MEN1KMT2A
SCHEMBL8176965 0.84 ESR1 (0.50) ESR1MEN1KMT2A
SCHEMBL8184744 0.83 CA1 (0.49) ESR1PDE5AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6130223-A Thienopyrimidine with phosphodiesterase V inhibiting effect MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-10-10 US disclosed