SCHEMBL5814645

SCHEMBL5814645

COc1ccc(CNc2nc(-c3ccncc3)nc3scc(C)c23)cc1Cl.Cc1csc2nc(-c3ccncc3)nc(Cl)c12

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.46
PDE5A O76074 11/20 0.43
ALDH1A1 P00352 1/20 0.42
HPGD P15428 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
BCDIN3D Q7Z5W3 2/20 0.42
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
PRKCI P41743 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5115035 0.96 ESR1 (0.48) ESR1PDE5ABCDIN3DMEN1KMT2A
SCHEMBL7522368 0.94 ALDH1A1 (0.47) ESR1ALDH1A1HPGDSMN1; SMN2MEN1
SCHEMBL7516802 0.91 ALDH1A1 (0.56) ESR1PDE5AALDH1A1HPGDSMN1; SMN2
SCHEMBL5119865 0.88 MEN1 (0.52) ESR1ALDH1A1MEN1KMT2APRKCI
SCHEMBL5122543 0.87 ALDH1A1 (0.52) ESR1PDE5AALDH1A1HPGDSMN1; SMN2
SCHEMBL7512225 0.86 NPC1 (0.44) ESR1PDE5AHPGDSMN1; SMN2BCDIN3D
SCHEMBL5120732 0.86 ESR1 (0.53) ESR1PRKCI
SCHEMBL8171015 0.85 ESR1 (0.47) ESR1PDE5ABCDIN3DMEN1KMT2A
SCHEMBL8169472 0.85 ESR1 (0.47) ESR1PDE5ABCDIN3DMEN1KMT2A
SCHEMBL5809020 0.84 ALDH1A1 (0.61) ESR1PDE5AALDH1A1HPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1685136-A1 USE OF THIENOPYRIMIDINES MERCK PATENT GmbH (DE) 2006-08-02 EP disclosed
WO-2005047292-A1 USE OF THIENOPYRIMIDINES MERCK PATENT GMBH (DE) 2005-05-26 WO disclosed