SCHEMBL8169668

SCHEMBL8169668

O=C(CBr)c1ccc(CN2C(=O)c3ccccc3C2=O)s1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 2/20 0.45
MAPK1 P28482 1/20 0.43
POLB P06746 2/20 0.43
HPGD P15428 1/20 0.43
CA12 O43570 1/20 0.41
CA9 Q16790 1/20 0.41
KMT2A Q03164 3/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC7 Q8WUI4 1/20 0.40
CASP3 P42574 1/20 0.39
MAPT P10636 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
MEN1 O00255 2/20 0.38
ALDH1A1 P00352 1/20 0.38
PKM P14618 1/20 0.38
GLA P06280 1/20 0.37
BRCA1 P38398 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11210405 0.86 MAPK1 (0.46) MAPK1POLBHPGDCA12CA9
SCHEMBL11212616 0.80 MAPK1 (0.44) MAPK1POLBHPGDCA12CA9
SCHEMBL6981532 0.79 CASP3 (0.45) MAPK1CA12CA9KMT2ACASP3
SCHEMBL13141314 0.76 MAPK1 (0.46) MAPK1POLBHPGDCA12CA9
SCHEMBL8422024 0.75 MAPK1 (0.46) MAPK1POLBHPGDCA12CA9
SCHEMBL8218019 0.72 CASP3 (0.49) MAPK1CA12CA9KMT2AHDAC1
SCHEMBL10505505 0.72 GRM5 (0.45) GSK3BCA12CA9KMT2AHDAC1
SCHEMBL31284533 0.71 GSK3B (0.60) GSK3BPOLBHPGDKMT2AMAPT
SCHEMBL5642365 0.71 CASP3 (0.44) MAPK1CA12CA9KMT2ACASP3
SCHEMBL2245062 0.70 GSK3B (0.58) GSK3BPOLBHPGDKMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6090804-A PSYCHOLOGICAL DISORDERS; SCHIZOPHRENIA THERAPY YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 2000-07-18 US disclosed
EP-0921123-A1 NOVEL THIOPHENE DERIVATIVES AND DRUG COMPOSITIONS CONTAINING THE SAME YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1999-06-09 EP disclosed