SCHEMBL8170605

SCHEMBL8170605

CC(C)OP(=O)(O)C(Cc1ccccn1)P(=O)(O)OC(C)C

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FDPS P14324 3/20 0.65
PTPRA P18433 1/20 0.45
PGR P06401 1/20 0.40
ADORA3 P0DMS8 1/20 0.40
PTGS1 P23219 1/20 0.40
SLC6A2 P23975 1/20 0.40
CYP1A2 P05177 2/20 0.40
CYP2D6 P10635 1/20 0.40
MAPT P10636 1/20 0.40
TSHR P16473 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
ALDH1A1 P00352 2/20 0.40
GRIN2D O15399 1/20 0.40
GRIN3B O60391 1/20 0.40
GRIN1 Q05586 1/20 0.40
GRIN2A Q12879 1/20 0.40
GRIN2B Q13224 1/20 0.40
GRIN2C Q14957 1/20 0.40
GRIN3A Q8TCU5 1/20 0.40
KCNA5 P22460 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8165506 0.94 FDPS (0.70) FDPSPTPRAPGRADORA3PTGS1
SCHEMBL8167468 0.85 FDPS (0.59) FDPSPTPRAALDH1A1GRIN2DGRIN3B
SCHEMBL8167866 0.85 FDPS (0.69) FDPSPTPRAALDH1A1GRIN2DGRIN3B
SCHEMBL8166906 0.81 FDPS (0.63) FDPSPTPRAPGRADORA3PTGS1
Piridronic Acid SCHEMBL223779 0.79 FDPS (1.00) FDPSPTPRASMN1; SMN2ALDH1A1GRIN2D
SCHEMBL10748069 0.78 FDPS (0.48) FDPSPTPRAPGRADORA3PTGS1
SCHEMBL8165637 0.74 FDPS (0.64) FDPSPTPRAPGRADORA3PTGS1
Piridronic Acid SCHEMBL634964 0.73 FDPS (0.79) FDPSPTPRASMN1; SMN2ALDH1A1GRIN2D
SCHEMBL8166214 0.72 FDPS (0.66) FDPS
SCHEMBL8168934 0.72 FDPS (0.69) FDPSCYP1A2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0563107-B1 NOVEL METHYLENEBISPHOSPHONIC ACID DERIVATIVES LEIRAS OY (FI) 2000-05-03 EP disclosed
US-5393748-A Treating bone disorders, Paget* s disease, calcium metabolism disorders LEIRAS OY (FI) 1995-02-28 US disclosed
EP-0563107-A1 NOVEL METHYLENEBISPHOSPHONIC ACID DERIVATIVES LEIRAS OY (FI) 1993-10-06 EP disclosed
WO-1992011269-A1 NOVEL METHYLENEBISPHOSPHONIC ACID DERIVATIVES LEIRAS OY (FI) 1992-07-09 WO disclosed