SCHEMBL8175404

SCHEMBL8175404

COc1ccc(NC(=O)NCc2ccccc2)cc1

nearest known ligand 0.89

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 6/20 0.89
NPC1 O15118 6/20 0.89
SMN1; SMN2 Q16637 2/20 0.76
HIF1A Q16665 1/20 0.70
MAOB P27338 1/20 0.69
HDAC1 Q13547 1/20 0.69
HDAC6 Q9UBN7 1/20 0.69
MEN1 O00255 2/20 0.67
KMT2A Q03164 2/20 0.67
CA2 P00918 1/20 0.67
HTT P42858 1/20 0.67
L3MBTL1 Q9Y468 1/20 0.66
FPR2 P25090 1/20 0.66
POLB P06746 1/20 0.66
MAPT P10636 3/20 0.65
NAMPT P43490 3/20 0.64
ALDH1A1 P00352 1/20 0.64
CASR P41180 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5427744 0.94 NPC1 (1.00) RAB9ANPC1SMN1; SMN2HIF1AMAOB
SCHEMBL17916794 0.92 SMN1; SMN2 (0.88) RAB9ANPC1SMN1; SMN2HIF1AHDAC1
SCHEMBL17831080 0.92 NPC1 (0.84) RAB9ANPC1SMN1; SMN2HIF1AMAOB
SCHEMBL23747763 0.91 NPC1 (0.78) RAB9ANPC1SMN1; SMN2HIF1AMAOB
SCHEMBL26097972 0.91 NPC1 (0.80) RAB9ANPC1SMN1; SMN2HIF1AMAOB
SCHEMBL26101164 0.89 NPC1 (0.80) RAB9ANPC1SMN1; SMN2HIF1AHDAC1
SCHEMBL23747796 0.89 NPC1 (0.74) RAB9ANPC1SMN1; SMN2HIF1AMAOB
SCHEMBL16562080 0.87 NPC1 (0.77) RAB9ANPC1SMN1; SMN2HIF1AMEN1
SCHEMBL23728269 0.87 POLB (0.81) RAB9ANPC1SMN1; SMN2HIF1AHDAC1
SCHEMBL23728200 0.87 NPC1 (0.77) RAB9ANPC1SMN1; SMN2HIF1AHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103664704-B A kind of synthetic N, the method for N '-disubstituted urea NANJING UNIVERSITY OF SCIENCE AND TECHNOLOGY (CN) 2016-05-18 CN disclosed
CN-105481723-A Preparation method for alkyl/benzyl/aryl urea compounds through heterogeneous-phase catalysis UNIV CHINA AGRICULTURAL 2016-04-13 CN disclosed
CN-103664704-A Method for synthesizing N,N'-disubstituent urea UNIV NANJING SCIENCE & TECH 2014-03-26 CN disclosed
US-6124288-A Xanthines and their therapeutic use DARWIN DISCOVERY, LTD. (GB) 2000-09-26 US disclosed
US-5821366-A Xanthines and their therapeutic use CHIROSCIENCE LIMITED (GB) 1998-10-13 US disclosed