SCHEMBL8178378

SCHEMBL8178378

CCNc1cccc(CNc2nc(-c3ccc(C(=O)O)cc3)nc3scc(C)c23)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.44
CYP1A2 P05177 3/20 0.44
CYP2D6 P10635 3/20 0.44
TSHR P16473 3/20 0.44
CYP2C19 P33261 3/20 0.44
HPGD P15428 2/20 0.44
MAPT P10636 2/20 0.44
ALOX15 P16050 1/20 0.44
HIF1A Q16665 1/20 0.44
HSD17B10 Q99714 1/20 0.44
ESR1 P03372 2/20 0.42
RXRA P19793 2/20 0.39
NR4A2 P43354 2/20 0.39
PDE4B Q07343 2/20 0.39
PDE4D Q08499 2/20 0.39
USP2 O75604 2/20 0.38
CYP3A4 P08684 2/20 0.38
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8169965 0.88 ESR1 (0.51) LMNACYP1A2CYP2D6TSHRCYP2C19
SCHEMBL8179470 0.87 ESR1 (0.45) LMNACYP1A2CYP2D6TSHRCYP2C19
SCHEMBL8171257 0.84 PDE5A (0.53) LMNACYP1A2CYP2D6TSHRCYP2C19
SCHEMBL8177939 0.82 ESR1 (0.51) LMNACYP1A2CYP2D6TSHRCYP2C19
SCHEMBL8170405 0.82 ESR1 (0.52) LMNACYP1A2CYP2D6TSHRCYP2C19
SCHEMBL8171050 0.81 KMT2A (0.50) LMNAMAPTESR1MEN1ALDH1A1
SCHEMBL8177979 0.80 PDE5A (0.45) HPGDESR1KDM4EMEN1ALDH1A1
SCHEMBL8184744 0.79 CA1 (0.49) LMNACYP1A2CYP2D6TSHRCYP2C19
SCHEMBL8171015 0.79 ESR1 (0.47) ESR1PDE4BPDE4DMEN1KMT2A
SCHEMBL8180832 0.76 PDE5A (0.50) LMNACYP1A2CYP2D6TSHRCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6130223-A Thienopyrimidine with phosphodiesterase V inhibiting effect MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-10-10 US disclosed