SCHEMBL8170405

SCHEMBL8170405

Cc1csc2nc(-c3ccc(C(=O)O)cc3)nc(NCc3ccc(F)cc3)c12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.52
PTGS2 P35354 2/20 0.44
KMT2A Q03164 2/20 0.43
LMNA P02545 2/20 0.43
MEN1 O00255 1/20 0.43
MAPT P10636 1/20 0.43
PPARA Q07869 1/20 0.43
CTNNB1 P35222 4/20 0.42
TCF7L2 Q9NQB0 4/20 0.42
F2 P00734 3/20 0.42
RAB9A P51151 1/20 0.42
USP2 O75604 2/20 0.41
TSHR P16473 2/20 0.41
HSD17B10 Q99714 1/20 0.41
VCP P55072 1/20 0.40
CYP1A2 P05177 2/20 0.40
CYP3A4 P08684 2/20 0.40
CYP2D6 P10635 2/20 0.40
HPGD P15428 2/20 0.40
CYP2C19 P33261 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8169965 0.92 ESR1 (0.51) ESR1PTGS2KMT2ALMNAMEN1
SCHEMBL8176965 0.90 ESR1 (0.50) ESR1PTGS2KMT2ALMNAMEN1
SCHEMBL8177939 0.86 ESR1 (0.51) ESR1KMT2ALMNAMEN1MAPT
SCHEMBL5129882 0.86 ESR1 (0.54) ESR1PTGS2KMT2ALMNAMEN1
SCHEMBL8171050 0.84 KMT2A (0.50) ESR1KMT2ALMNAMEN1MAPT
SCHEMBL8184718 0.83 FLT3 (0.51) PTGS2KMT2ALMNAMEN1MAPT
SCHEMBL8179470 0.83 ESR1 (0.45) ESR1LMNAMAPTUSP2TSHR
SCHEMBL8184744 0.82 CA1 (0.49) ESR1KMT2ALMNAMEN1MAPT
SCHEMBL8171015 0.82 ESR1 (0.47) ESR1KMT2AMEN1
SCHEMBL8178378 0.82 LMNA (0.44) ESR1KMT2ALMNAMEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6130223-A Thienopyrimidine with phosphodiesterase V inhibiting effect MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-10-10 US disclosed