SCHEMBL8178795

SCHEMBL8178795

CC(C)C(=O)Nc1c(N)nc(S)nc1O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.40
MDM4 O15151 1/20 0.37
TP53 P04637 1/20 0.37
ALDH1A1 P00352 3/20 0.36
LMNA P02545 2/20 0.36
HSD17B10 Q99714 2/20 0.36
TYR P14679 1/20 0.33
GAA P10253 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
MAPT P10636 1/20 0.33
KDM4E B2RXH2 2/20 0.32
CA1 P00915 2/20 0.32
CA2 P00918 2/20 0.32
CA9 Q16790 2/20 0.32
CA4 P22748 1/20 0.32
ADORA1 P30542 1/20 0.32
TSHR P16473 2/20 0.32
SCN10A Q9Y5Y9 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8166609 0.72 NPSR1 (0.37) NPSR1MDM4TP53ALDH1A1LMNA
SCHEMBL15565552 0.67 KMT2A (0.41) ALDH1A1LMNAHSD17B10CYP1A2MAPT
SCHEMBL10205212 0.64 LMNA (0.31) LMNA
SCHEMBL739774 0.64
SCHEMBL3804852 0.63 KMT2A (0.38) ALDH1A1LMNAHSD17B10GAACYP1A2
SCHEMBL10995388 0.62 ADORA1 (0.42) TP53ALDH1A1LMNAHSD17B10CA1
SCHEMBL11015282 0.62 KMT2A (0.37) ALDH1A1GAATSHRKMT2A
SCHEMBL13540000 0.62 HPGD (0.33) ALDH1A1HSD17B10KDM4EHPGD
SCHEMBL16316425 0.62 ADORA1 (0.56) NPSR1MDM4TP53ALDH1A1LMNA
Hydrochloric Acid SCHEMBL4410483 0.62

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6057445-A FORMATION OF CARBON NITROGEN BOND, CYCLIZATION AND HALOGENATION EURO-CELTIQUE S.A. (LU) 2000-05-02 US disclosed
WO-1999031104-A1 PREPARATION OF 3-SUBSTITUTED ADENINES AND IMIDAZO PYRIDINES EURO-CELTIQUE, S.A. (LU) 1999-06-24 WO disclosed