SCHEMBL8179337

SCHEMBL8179337

Cc1sc2nc(C3CCC(C(=O)O)CC3)nc(NCc3ccc4c(c3)OCO4)c2c1C

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.48
PDE4A P27815 2/20 0.47
PDE4B Q07343 2/20 0.47
PDE4C Q08493 2/20 0.47
PDE4D Q08499 2/20 0.47
PTPN12 Q05209 1/20 0.47
PTPN22 Q9Y2R2 1/20 0.47
MAPT P10636 3/20 0.46
LMNA P02545 2/20 0.46
ALOX15 P16050 1/20 0.46
SMN1; SMN2 Q16637 5/20 0.46
CHRM4 P08173 3/20 0.43
RAB9A P51151 1/20 0.43
GAA P10253 2/20 0.42
POLB P06746 2/20 0.42
HTT P42858 2/20 0.42
MEN1 O00255 1/20 0.42
TP53 P04637 1/20 0.42
TSHR P16473 1/20 0.42
MAPK1 P28482 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8180824 0.92 ALDH1A1 (0.51) ALDH1A1PDE4APDE4BPDE4CPDE4D
SCHEMBL8179541 0.92 PDE4A (0.50) ALDH1A1PDE4APDE4BPDE4CPDE4D
Bicarbonate SCHEMBL7017359 0.90 PTPN12 (0.47) ALDH1A1PTPN12PTPN22MAPTLMNA
SCHEMBL8178383 0.86 ALDH1A1 (0.51) ALDH1A1PTPN12PTPN22MAPTLMNA
SCHEMBL8179485 0.86 ALDH1A1 (0.49) ALDH1A1PDE4APDE4BPDE4CPDE4D
SCHEMBL8177034 0.86 PDE4A (0.64) ALDH1A1PDE4APDE4BPDE4CPDE4D
SCHEMBL8183118 0.85 ALDH1A1 (0.59) ALDH1A1PDE4APDE4BPDE4CPDE4D
SCHEMBL8172347 0.85 PDE4A (0.52) ALDH1A1PDE4APDE4BPDE4CPDE4D
SCHEMBL8181994 0.85 ALDH1A1 (0.52) ALDH1A1PDE4APDE4BPDE4CPDE4D
SCHEMBL8184394 0.85 PTPN12 (0.64) ALDH1A1PDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6130223-A Thienopyrimidine with phosphodiesterase V inhibiting effect MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-10-10 US disclosed