SCHEMBL8190066

SCHEMBL8190066

CC(=O)OC[C@H]1O[C](C(F)(F)[C]2O[C@H](COC(C)=O)[C@@H](OC(C)=O)[C@H](OC(C)=O)[C@@H]2OC(C)=O)[C@@H](OC(C)=O)[C@@H](OC(C)=O)[C@@H]1OC(C)=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.44
THRB P10828 2/20 0.42
CYP2D6 P10635 1/20 0.42
HSD17B10 Q99714 1/20 0.42
NR3C1 P04150 1/20 0.41
FYN P06241 1/20 0.41
ADRA2A P08913 1/20 0.41
ADORA3 P0DMS8 1/20 0.41
ADRA2B P18089 1/20 0.41
DRD4 P21917 1/20 0.41
DRD3 P35462 1/20 0.41
CA12 O43570 13/20 0.41
CA1 P00915 13/20 0.41
CA2 P00918 13/20 0.41
CA4 P22748 8/20 0.41
CA5A P35218 8/20 0.41
CA7 P43166 8/20 0.41
CA5B Q9Y2D0 8/20 0.41
CA9 Q16790 7/20 0.40
PTPN1 P18031 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17794446 0.80 TSHR (0.48) TSHRTHRBCYP2D6HSD17B10NR3C1
SCHEMBL7151005 0.80 TSHR (0.48) TSHRTHRBCYP2D6HSD17B10NR3C1
SCHEMBL7155828 0.80 TSHR (0.48) TSHRTHRBCYP2D6HSD17B10NR3C1
SCHEMBL7152306 0.80 TSHR (0.48) TSHRTHRBCYP2D6HSD17B10NR3C1
SCHEMBL11778919 0.80 TSHR (0.48) TSHRTHRBCYP2D6HSD17B10NR3C1
SCHEMBL8197918 0.78 TSHR (0.47) TSHRTHRBCYP2D6HSD17B10NR3C1
SCHEMBL2588471 0.78 TSHR (0.47) TSHRTHRBCYP2D6HSD17B10NR3C1
SCHEMBL9694585 0.75 TSHR (0.46) TSHRTHRBCYP2D6HSD17B10NR3C1
SCHEMBL6239338 0.75 TSHR (0.46) TSHRTHRBCYP2D6HSD17B10NR3C1
SCHEMBL11167401 0.71 THRB (0.64) TSHRTHRBCYP2D6HSD17B10NR3C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0934325-A4 TETRAPHOSPHONATE BICYCLIC TRISANHYDRIDES PHARMASSET LTD (US) 2000-08-16 EP disclosed
EP-0934325-A1 TETRAPHOSPHONATE BICYCLIC TRISANHYDRIDES Pharmasset, Ltd. (US) 1999-08-11 EP disclosed
WO-1998015563-A1 TETRAPHOSPHONATE BICYCLIC TRISANHYDRIDES PHARMASSET, LTD. (US) 1998-04-16 WO disclosed