SCHEMBL8192147

SCHEMBL8192147

C#CCNC(=O)c1c(NCC(=O)O)nc(C#Cc2ccc(OC)c(OC)c2)n1C

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 2/20 0.35
ACACB O00763 2/20 0.35
CFTR P13569 3/20 0.34
FLT1 P17948 2/20 0.34
KDR P35968 2/20 0.34
TP53 P04637 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
KDM4E B2RXH2 3/20 0.33
POLB P06746 2/20 0.32
ALDH1A1 P00352 2/20 0.32
GAA P10253 2/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
RIPK1 Q13546 1/20 0.32
PDE4A P27815 1/20 0.32
PDE4B Q07343 1/20 0.32
PDE4C Q08493 1/20 0.32
PDE4D Q08499 1/20 0.32
LMNA P02545 1/20 0.32
HPGD P15428 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8183622 0.93 ACACB (0.37) ACACBCFTRFLT1KDRTP53
SCHEMBL8184881 0.91 ACACB (0.35) ACACBCFTRFLT1KDRTP53
SCHEMBL8175218 0.91 ACACB (0.36) ACACBCFTRFLT1KDRTP53
SCHEMBL8189038 0.91 PGK1 (0.38) ACACBCFTRFLT1KDRTP53
SCHEMBL8179729 0.90 ACACB (0.35) ACACBCFTRFLT1KDRTP53
SCHEMBL8184729 0.89 CFTR (0.35) ACACBCFTRFLT1KDRKDM4E
SCHEMBL8180999 0.89 SYK (0.39) ACACBCFTRFLT1KDRTP53
SCHEMBL8179960 0.89 TNF (0.37) ACACBCFTRFLT1KDRSMN1; SMN2
SCHEMBL8184731 0.88 ACACB (0.38) ACACBCFTRFLT1KDRTP53
SCHEMBL8175450 0.88 CFTR (0.35) ACACBCFTRFLT1KDRTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008077557-A1 8-ETHINYLXANTHINE DERIVATIVES AS SELECTIVE A2A RECEPTOR ANTAGONISTS SCHWARZ PHARMA AG (DE) 2008-07-03 WO disclosed