SCHEMBL8196255

SCHEMBL8196255

CCC[C@@H](CNCCc1ccccn1)NC(=O)C1CO1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.48
CYP1A2 P05177 2/20 0.48
CYP2C19 P33261 2/20 0.48
HSD11B1 P28845 1/20 0.41
LMNA P02545 2/20 0.39
TDP1 Q9NUW8 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
TAAR1 Q96RJ0 1/20 0.38
ALOX15 P16050 1/20 0.38
DPP7 Q9UHL4 1/20 0.38
TAS1R3 Q7RTX0 2/20 0.38
TAS1R1 Q7RTX1 2/20 0.38
HPGD P15428 1/20 0.38
TSHR P16473 1/20 0.38
MAPK1 P28482 1/20 0.38
CYP2D6 P10635 2/20 0.37
KDM4E B2RXH2 2/20 0.37
GAA P10253 1/20 0.37
POLB P06746 1/20 0.37
FPR3 P25089 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8202246 0.82 KMT2A (0.50) ALDH1A1CYP1A2CYP2C19HSD11B1TAS1R3
SCHEMBL8204207 0.81 ALDH1A1 (0.43) ALDH1A1CYP1A2CYP2C19HSD11B1LMNA
SCHEMBL8203636 0.77 CYP1A2 (0.62) ALDH1A1CYP1A2CYP2C19LMNATDP1
SCHEMBL31690650 0.73 SMN1; SMN2 (0.58) ALDH1A1CYP1A2CYP2C19HSD11B1LMNA
SCHEMBL15318323 0.67 CYP1A2 (0.77) ALDH1A1CYP1A2CYP2C19LMNATDP1
SCHEMBL3422911 0.67 ALDH1A1 (1.00) ALDH1A1CYP1A2CYP2C19LMNATDP1
SCHEMBL6752172 0.67 CYP1A2 (0.65) ALDH1A1CYP1A2CYP2C19LMNATDP1
SCHEMBL8208537 0.65 KMT2A (0.53) ALDH1A1CYP1A2CYP2C19LMNATDP1
SCHEMBL746674 0.65 CYP1A2 (0.67) ALDH1A1CYP1A2CYP2C19LMNATDP1
SCHEMBL13995588 0.65 CYP1A2 (0.77) ALDH1A1CYP1A2CYP2C19LMNATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008042480-A2 EPOXIDE INHIBITORS OF CYSTEINE PROTEASES THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2008-04-10 WO disclosed