SCHEMBL8197486

SCHEMBL8197486

Cc1nc2c(s1)C(=O)NCCC2

nearest known ligand 0.67

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.61
TSHR P16473 2/20 0.54
GRM5 P41594 6/20 0.41
CDK1 P06493 1/20 0.37
MAPKAPK2 P49137 1/20 0.37
ATAD2 Q6PL18 1/20 0.36
MAPK1 P28482 2/20 0.36
USP2 O75604 1/20 0.36
HTT P42858 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
OR51E2 Q9H255 1/20 0.34
OGA O60502 2/20 0.33
GAA P10253 1/20 0.33
GFER P55789 1/20 0.33
KDM4E B2RXH2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4409177 0.89 GRM5 (0.50) ALDH1A1TSHRGRM5ATAD2HTT
SCHEMBL12938272 0.82 ALDH1A1 (0.57) ALDH1A1TSHRGRM5CDK1MAPKAPK2
SCHEMBL12938269 0.81 ALDH1A1 (0.59) ALDH1A1TSHRGRM5CDK1MAPKAPK2
SCHEMBL2073986 0.81 ALDH1A1 (0.56) ALDH1A1TSHRGRM5CDK1MAPKAPK2
SCHEMBL3587356 0.76 ALDH1A1 (0.51) ALDH1A1TSHRGRM5MAPK1USP2
SCHEMBL19152800 0.76 ALDH1A1 (0.36) ALDH1A1TSHR
SCHEMBL6118325 0.76 ALDH1A1 (0.56) ALDH1A1TSHRGRM5CDK1MAPK1
SCHEMBL2035154 0.76 ALDH1A1 (0.61) ALDH1A1TSHRGRM5CDK1MAPK1
SCHEMBL303576 0.71 PIK3CD (0.67) ALDH1A1TSHRHTTOGA
SCHEMBL15001035 0.71 CCNE1 (0.41) ALDH1A1CDK1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000064904-A1 5,7-BICYCLIC AMIDINE DERIVATIVES USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS ASTRAZENECA AB (SE) 2000-11-02 WO disclosed