SCHEMBL8197962

SCHEMBL8197962

CCCn1c(=O)nc(-c2cccc(Cl)c2)c2ccc(C)nc21

nearest known ligand 0.64

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.64
CYP1A2 P05177 3/20 0.64
CYP2C9 P11712 3/20 0.64
ALDH1A1 P00352 2/20 0.64
HSD17B10 Q99714 2/20 0.64
CYP3A4 P08684 1/20 0.64
TSHR P16473 1/20 0.64
LMNA P02545 1/20 0.47
GAA P10253 1/20 0.47
HPGD P15428 1/20 0.47
HTT P42858 1/20 0.47
ADORA1 P30542 1/20 0.45
MAOB P27338 1/20 0.42
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42
CYP2C19 P33261 1/20 0.42
DPP4 P27487 1/20 0.41
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8193560 0.91 KDM4E (0.77) KDM4ECYP1A2CYP2C9ALDH1A1HSD17B10
SCHEMBL8193126 0.88 ALDH1A1 (0.49) KDM4ECYP1A2CYP2C9ALDH1A1HSD17B10
SCHEMBL8224986 0.85 KDM4E (0.69) KDM4ECYP1A2CYP2C9ALDH1A1HSD17B10
SCHEMBL8198547 0.84 KDM4E (0.58) KDM4ECYP1A2CYP2C9ALDH1A1HSD17B10
SCHEMBL8192913 0.79 ALDH1A1 (0.57) KDM4ECYP1A2CYP2C9ALDH1A1HSD17B10
SCHEMBL8183814 0.79 KDM4E (0.60) KDM4ECYP1A2CYP2C9ALDH1A1HSD17B10
SCHEMBL157252 0.78 ALDH1A1 (1.00) KDM4ECYP1A2CYP2C9ALDH1A1HSD17B10
SCHEMBL8183859 0.78 ALDH1A1 (0.76) KDM4ECYP1A2CYP2C9ALDH1A1HSD17B10
SCHEMBL29372580 0.78 ALDH1A1 (1.00) KDM4ECYP1A2CYP2C9ALDH1A1HSD17B10
SCHEMBL8192931 0.77 ALDH1A1 (0.57) KDM4ECYP1A2CYP2C9ALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6136810-A DRUGS AS ENZYME INHIBITORS OF PHOSPHODIESTERASE YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 2000-10-24 US disclosed
EP-0885894-A1 PYRIDO [2,3-D] PYRIMIDINE DERIVATIVES AND MEDICINAL COMPOSITIONS THEREOF YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1998-12-23 EP disclosed