SCHEMBL8198030

SCHEMBL8198030

CCc1ccc(Cl)c(N(C(=N)NC)c2cccc(C(F)(F)F)c2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 7/20 0.48
LMNA P02545 3/20 0.37
MAPT P10636 2/20 0.37
ADRA2C P18825 1/20 0.37
HTR2A P28223 1/20 0.37
SLC6A4 P31645 1/20 0.37
ADRA1A P35348 1/20 0.37
DRD3 P35462 1/20 0.37
OPRK1 P41145 1/20 0.37
HTR2B P41595 1/20 0.37
CETP P11597 3/20 0.37
HPGD P15428 1/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
THRB P10828 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.34
CYP2D6 P10635 2/20 0.34
CYP2C19 P33261 2/20 0.34
PLA2G1B P04054 1/20 0.34
CYP1A2 P05177 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8397630 0.87 SIGMAR1 (0.50) SIGMAR1HTR2AHTR2BCETPMEN1
SCHEMBL8332178 0.81 SIGMAR1 (0.63) SIGMAR1
SCHEMBL8198033 0.80 SIGMAR1 (0.46) SIGMAR1
SCHEMBL6719420 0.76 SIGMAR1 (0.48) SIGMAR1MEN1KMT2ACYP2D6CYP2C19
SCHEMBL6727687 0.76 SIGMAR1 (0.51) SIGMAR1LMNAMAPTHPGDMEN1
Hydrochloric Acid SCHEMBL7201876 0.75 SIGMAR1 (0.49) SIGMAR1CYP2D6CYP2C19CYP1A2
SCHEMBL27498292 0.73 SIGMAR1 (0.64) SIGMAR1
SCHEMBL8401133 0.72 SIGMAR1 (0.40) SIGMAR1MAPTCETPHPGDGAA
SCHEMBL27482600 0.72 SIGMAR1 (0.59) SIGMAR1SLC6A4CYP2D6CYP3A4
SCHEMBL27519224 0.71 SIGMAR1 (0.53) SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6156741-A Therapeutic substituted guanidines CAMBRIDGE NEUROSCIENCE, INC. (US) 2000-12-05 US claimed