SCHEMBL8199526

SCHEMBL8199526

O=C1c2ccc(OCc3cccnc3)cc2CCC1CCN1CCC(c2ccccc2)CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1D P25100 1/20 0.49
ADRA1A P35348 1/20 0.49
ADRA1B P35368 1/20 0.49
DRD2 P14416 4/20 0.45
HTR2A P28223 4/20 0.45
HTR2C P28335 4/20 0.45
HTR2B P41595 3/20 0.45
SIGMAR1 Q99720 3/20 0.45
GPR84 Q9NQS5 1/20 0.45
CYP19A1 P11511 1/20 0.42
HTR7 P34969 1/20 0.42
PRMT5 O14744 1/20 0.42
WDR77 Q9BQA1 1/20 0.42
HRH3 Q9Y5N1 2/20 0.41
ITGB3 P05106 1/20 0.41
ITGA2B P08514 1/20 0.41
HTR1A P08908 1/20 0.41
TRPA1 O75762 1/20 0.40
CHRM4 P08173 1/20 0.40
CYP24A1 Q07973 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8198852 0.91 ADRA1D (0.57) ADRA1DADRA1AADRA1BDRD2HTR2A
SCHEMBL8199711 0.91 ADRA1D (0.53) ADRA1DADRA1AADRA1BDRD2HTR2A
SCHEMBL8200296 0.86 ADRA1D (0.50) ADRA1DADRA1AADRA1BDRD2HTR2A
SCHEMBL8200537 0.86 ADRA1D (0.56) ADRA1DADRA1AADRA1BDRD2HTR2A
SCHEMBL8192983 0.86 ADRA1D (0.49) ADRA1DADRA1AADRA1BDRD2HTR2A
SCHEMBL8199674 0.86 MAOB (0.50) ADRA1DADRA1AADRA1BDRD2HTR2A
SCHEMBL8199290 0.85 ADRA1D (0.55) ADRA1DADRA1AADRA1BDRD2HTR2A
SCHEMBL8192734 0.85 ADRA1D (0.55) ADRA1DADRA1AADRA1BDRD2HTR2A
SCHEMBL8192177 0.85 HTR2C (0.54) ADRA1DADRA1AADRA1BDRD2HTR2A
SCHEMBL6491492 0.84 ADRA1D (0.54) ADRA1DADRA1AADRA1BDRD2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6048877-A Tetralone derivatives as antiarrhythmic agents BRISTOL-MYERS SQUIBB COMPANY (US) 2000-04-11 US claimed
WO-1998036749-A1 TETRALONE DERIVATIVES AS ANTIARRHYTHMIC AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 1998-08-27 WO claimed
US-6048877-A Tetralone derivatives as antiarrhythmic agents BRISTOL-MYERS SQUIBB COMPANY (US) 2000-04-11 US disclosed