SCHEMBL8199675

SCHEMBL8199675

CC(C)CN(CC(C)C)C(=O)CC1CCc2cc(OCc3ccccc3)ccc2C1=O

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.56
ITGA2B P08514 1/20 0.56
CYP24A1 Q07973 6/20 0.47
CYP26A1 O43174 3/20 0.47
MAOB P27338 3/20 0.47
MAOA P21397 2/20 0.47
CYP27A1 Q02318 3/20 0.45
FFAR1 O14842 1/20 0.43
THRA P10827 1/20 0.43
THRB P10828 1/20 0.43
CYP19A1 P11511 1/20 0.42
HRH3 Q9Y5N1 2/20 0.41
GRIN1 Q05586 1/20 0.41
GRIN2B Q13224 1/20 0.41
S1PR1 P21453 1/20 0.41
NPC1 O15118 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
NFKB1 P19838 1/20 0.41
GRM5 P41594 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8203550 0.85 ITGB3 (0.58) ITGB3ITGA2BCYP24A1CYP26A1MAOB
SCHEMBL4622240 0.82 ITGB3 (0.59) ITGB3ITGA2BCYP24A1CYP26A1MAOB
SCHEMBL8198563 0.81 ITGB3 (0.54) ITGB3ITGA2BCYP24A1CYP26A1MAOB
SCHEMBL8200699 0.80 ITGB3 (0.55) ITGB3ITGA2BCYP24A1CYP26A1MAOB
SCHEMBL8198784 0.80 ITGB3 (0.55) ITGB3ITGA2BCYP24A1CYP26A1MAOB
SCHEMBL8198782 0.80 ITGB3 (0.55) ITGB3ITGA2BCYP24A1CYP26A1MAOB
SCHEMBL8200056 0.80 ITGB3 (0.54) ITGB3ITGA2BCYP24A1CYP26A1MAOB
SCHEMBL8199287 0.79 MAOB (0.51) ITGB3ITGA2BCYP24A1CYP26A1MAOB
SCHEMBL8200304 0.79 ITGB3 (0.60) ITGB3ITGA2BCYP24A1CYP26A1MAOB
SCHEMBL8204211 0.78 ITGB3 (0.57) ITGB3ITGA2BCYP24A1CYP26A1MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998036749-A1 TETRALONE DERIVATIVES AS ANTIARRHYTHMIC AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 1998-08-27 WO claimed
US-6048877-A Tetralone derivatives as antiarrhythmic agents BRISTOL-MYERS SQUIBB COMPANY (US) 2000-04-11 US disclosed