SCHEMBL8199890

SCHEMBL8199890

CCOP(=O)(OCC)C(C)C(=O)Cl

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.44
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
TP53 P04637 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
POLB P06746 1/20 0.39
TSHR P16473 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.37
MAPT P10636 2/20 0.36
PPARD Q03181 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL319717 0.80 TSHR (0.42) GAACYP3A4CYP2C9CYP2C19TP53
SCHEMBL4050 0.80 POLB (0.44) GAACYP3A4CYP2C9CYP2C19TP53
SCHEMBL16814501 0.79 GAA (0.41) GAACYP3A4CYP2C9CYP2C19TP53
SCHEMBL9445952 0.78 GAA (0.40) GAACYP3A4CYP2C9CYP2C19TP53
SCHEMBL5839781 0.78 GAA (0.40) GAACYP3A4CYP2C9CYP2C19TP53
SCHEMBL24165690 0.78 CYP3A4 (0.47) GAACYP3A4CYP2C9CYP2C19TP53
SCHEMBL10108 0.78 GAA (0.40) GAACYP3A4CYP2C9CYP2C19TP53
SCHEMBL13847695 0.77 CYP3A4 (0.42) GAACYP3A4CYP2C9CYP2C19TP53
SCHEMBL14671697 0.77 CYP3A4 (0.42) GAACYP3A4CYP2C9CYP2C19TP53
SCHEMBL4098271 0.77 CYP3A4 (0.42) GAACYP3A4CYP2C9CYP2C19TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015088564-A1 P2X4 RECEPTOR MODULATING COMPOUNDS SUNOVION PHARMACEUTICALS INC. (US) 2015-06-18 WO disclosed
US-20090036638-A1 Contrast Dyes for Inkjet Lithographic Printing Plates AGFA GRAPHICS NV (BE) 2009-02-05 US disclosed
US-20080280055-A1 Inkjet Lithographic Printing Plates and Method for Their Preparation AGFA GRAPHICS NV (BE) 2008-11-13 US disclosed
EP-0783504-B1 [1,2,4]TRIAZOLO[4,3-a]QUINOXALINONE DERIVATIVES, THEIR PREPARATION AND USE AS ANTAGONISTS OF AMPA-RECEPTORS NOVO NORDISK AS (DK) 2000-03-15 EP disclosed
US-6001832-A [1,2,4]triazolo[4,3-a]quinoxalinone derivatives, their preparation and use NOVO NORDISKALS (DK) 1999-12-14 US disclosed
EP-0783504-A1 [1,2,4]TRIAZOLO[4,3-a]QUINOXALINONE DERIVATIVES, THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1997-07-16 EP disclosed
WO-1996008492-A1 [1,2,4]TRIAZOLO[4,3-a]QUINOXALINONE DERIVATIVES, THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1996-03-21 WO disclosed