SCHEMBL8200370

SCHEMBL8200370

COc1ccccc1-c1nn2ccccc2c1-c1ccc(=O)n(C)n1

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 2/20 0.44
BRD4 O60885 2/20 0.44
ADORA2A P29274 1/20 0.38
MAPK1 P28482 1/20 0.37
MAPK14 Q16539 1/20 0.37
JAK2 O60674 1/20 0.37
PDE5A O76074 1/20 0.37
PDE3A Q14432 1/20 0.37
ALDH1A1 P00352 2/20 0.36
IGF1R P08069 1/20 0.35
GRM2 Q14416 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8197666 0.84 ADORA1 (0.48) ADORA1BRD4MAPK1PDE5APDE3A
SCHEMBL8193833 0.82 ADORA1 (0.52) ADORA1ADORA2AMAPK1MAPK14ALDH1A1
SCHEMBL8186528 0.81 PDE3A (0.60) ADORA1ADORA2AMAPK1MAPK14JAK2
SCHEMBL8809138 0.81 ADORA1 (0.64) ADORA1BRD4ADORA2AMAPK1MAPK14
SCHEMBL7658127 0.76 ADORA1 (0.53) ADORA1ADORA2AMAPK1MAPK14IGF1R
SCHEMBL6824871 0.75 NPC1 (0.38) ADORA1BRD4ADORA2AALDH1A1
SCHEMBL7364069 0.74 PDE1A (0.39) ADORA1BRD4ADORA2AMAPK14ALDH1A1
SCHEMBL6822006 0.72 ADORA1 (0.46) ADORA1BRD4MAPK1IGF1R
SCHEMBL7036909 0.71 ADORA1 (0.43) ADORA1BRD4ADORA2AMAPK1PDE5A
SCHEMBL7371668 0.71 ADORA2A (0.37) ADORA1BRD4ADORA2AMAPK14ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000024742-A1 PYRAZOLOPYRIDINE AS ADENOSINE ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-05-04 WO disclosed