SCHEMBL8200718

SCHEMBL8200718

CCC=Cc1ccccc1-c1ccc(C2=NCCN2)cc1

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 13/20 0.51
ALDH1A1 P00352 1/20 0.45
CYP1A2 P05177 1/20 0.45
HPGD P15428 1/20 0.45
CASP1 P29466 1/20 0.45
CASP7 P55210 1/20 0.45
HSD17B10 Q99714 1/20 0.45
HTR1D P28221 1/20 0.44
ADRA1A P35348 1/20 0.44
MAOA P21397 1/20 0.44
MAOB P27338 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8200716 1.00 NISCH (0.51) NISCHALDH1A1CYP1A2HPGDCASP1
SCHEMBL8194858 0.79 NISCH (0.58) NISCHHTR1DADRA1A
SCHEMBL8194859 0.79 NISCH (0.58) NISCHHTR1DADRA1A
SCHEMBL8201031 0.75 NISCH (0.54) NISCHALDH1A1CYP1A2HPGDCASP1
SCHEMBL8201034 0.75 NISCH (0.54) NISCHALDH1A1CYP1A2HPGDCASP1
SCHEMBL29287250 0.75 NOTUM (0.38) ALDH1A1CYP1A2HSD17B10
SCHEMBL1024642 0.75 BACE1 (0.43)
SCHEMBL1471407 0.75 BACE1 (0.43)
Alcohol SCHEMBL28563093 0.74 NISCH (0.79) NISCHALDH1A1CYP1A2HPGDCASP1
SCHEMBL3532943 0.72 NISCH (0.65) NISCHHTR1DADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000078726-A1 IMIDAZOLINE DERIVATIVES FOR THE TREATMENT OF DIABETES, ESPECIALLY TYPE II DIABETES ELI LILLY AND COMPANY (US) 2000-12-28 WO disclosed