SCHEMBL8201330

SCHEMBL8201330

C=C(C)c1ccc(-n2nc(Cl)cc2-c2ccc([S+](C)[O-])cc2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.39
PPP1CA P62136 1/20 0.39
CHRNA7 P36544 1/20 0.38
MALT1 Q9UDY8 4/20 0.37
RPA1 P27694 3/20 0.37
NFKB1 P19838 1/20 0.37
NFKB2 Q00653 1/20 0.37
RELA Q04206 1/20 0.37
PTGS2 P35354 4/20 0.35
PTGS1 P23219 1/20 0.35
SMPD1 P17405 1/20 0.35
HDAC3 O15379 1/20 0.35
HDAC4 P56524 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC7 Q8WUI4 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC10 Q969S8 1/20 0.35
HDAC11 Q96DB2 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8188387 0.85 PTGS2 (0.49) SMN1; SMN2PPP1CACHRNA7MALT1RPA1
SCHEMBL8234603 0.79 CYP2C9 (0.40) SMN1; SMN2PPP1CACHRNA7MALT1RPA1
SCHEMBL8234607 0.78 CYP2C9 (0.41) SMN1; SMN2PPP1CACHRNA7MALT1RPA1
SCHEMBL8218313 0.77 PPP1CA (0.50) SMN1; SMN2PPP1CACHRNA7MALT1RPA1
SCHEMBL8188245 0.77 PTGS2 (0.44) SMN1; SMN2CHRNA7MALT1PTGS2CA1
SCHEMBL8260353 0.75 PTGS2 (0.43) SMN1; SMN2CHRNA7MALT1PTGS2CA1
SCHEMBL7471309 0.71 PTGS2 (0.57) PTGS2PTGS1HDAC3HDAC4HDAC1
SCHEMBL9055803 0.70 MEN1 (0.53) SMN1; SMN2PPP1CACHRNA7MALT1RPA1
SCHEMBL25149362 0.68 PTGS2 (0.68) PTGS2PTGS1HDAC3HDAC4HDAC1
SCHEMBL9205418 0.68 PTGS2 (0.52) CHRNA7MALT1PTGS2PTGS1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000018741-A2 PYRAZOLE COMPOUNDS AS COX-2 INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-06 WO claimed