SCHEMBL8201447

SCHEMBL8201447

C=C(Cl)CC(CC(=O)OC(C)(C)C)C(=O)O

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GRIK1 P39086 1/20 0.46
GRIK2 Q13002 1/20 0.46
MEN1 O00255 1/20 0.39
GAA P10253 1/20 0.39
KMT2A Q03164 1/20 0.39
CYP2D6 P10635 1/20 0.36
HDAC3 O15379 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
CA2 P00918 1/20 0.32
CA9 Q16790 1/20 0.32
SLC15A1 P46059 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8201450 1.00 GRIK1 (0.46) GRIK1GRIK2MEN1GAAKMT2A
SCHEMBL4839844 0.87 MEN1 (0.47) MEN1GAAKMT2ACYP2D6HDAC3
SCHEMBL8204183 0.83 CYP2D6 (0.38) GRIK1GRIK2MEN1GAAKMT2A
SCHEMBL8204187 0.83 CYP2D6 (0.38) GRIK1GRIK2MEN1GAAKMT2A
SCHEMBL8192995 0.83 MEN1 (0.39) MEN1GAAKMT2ACYP2D6HDAC3
SCHEMBL8192997 0.83 MEN1 (0.39) MEN1GAAKMT2ACYP2D6HDAC3
SCHEMBL4755353 0.78 CA2 (0.45) MEN1GAAKMT2ACYP2D6HDAC3
SCHEMBL12268130 0.78 CA2 (0.45) MEN1GAAKMT2ACYP2D6HDAC3
SCHEMBL12047679 0.78 MEN1 (0.43) MEN1GAAKMT2ACYP2D6HDAC3
SCHEMBL4831221 0.77 GAA (0.40) MEN1GAAKMT2ACYP2D6HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0882138-B1 STEREOSELECTIVE PREPARATION OF 2-SUBSTITUTED SUCCINIC DERIVATIVES BOEHRINGER INGELHEIM CA LTD (CA) 2000-07-05 EP disclosed
US-5808085-A CHEMICAL INTERMEDIATES FOR RENIN INHIBITING COMPOUNDS BOEHRINGER INGELHEIM (CANADA) LTD. (CA) 1998-09-15 US disclosed