SCHEMBL8201772

SCHEMBL8201772

CC(C)(C(=O)NCC(F)(F)C(F)(F)F)C(=O)N[C@H]1CN(C(=O)O)c2ccccc2N(CC(F)(F)F)C1=O

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PSEN1 P49768 2/20 0.42
PSEN2 P49810 2/20 0.42
APH1B Q8WW43 2/20 0.42
NCSTN Q92542 2/20 0.42
APH1A Q96BI3 2/20 0.42
PSENEN Q9NZ42 2/20 0.42
SCN9A Q15858 11/20 0.41
XIAP P98170 7/20 0.41
CYP3A4 P08684 5/20 0.41
SCN10A Q9Y5Y9 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8209811 0.92 SCN9A (0.41) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL14093728 0.89 PSEN1 (0.40) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL4434451 0.84 PSEN1 (0.43) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL5541816 0.84 PSEN1 (0.43) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL4434392 0.84 XIAP (0.49) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL4434389 0.84 XIAP (0.49) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL8216655 0.81 SCN9A (0.39) SCN9AXIAPCYP3A4SCN10A
SCHEMBL14093717 0.81 SCN9A (0.39) SCN9AXIAPCYP3A4SCN10A
SCHEMBL5014049 0.78 SCN9A (0.43) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL8207632 0.78 SCN9A (0.43) PSEN1PSEN2APH1BNCSTNAPH1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008034735-A2 4-OXO-2,3,4,5-TETRAHYDRO-BENZO[B][1,4]DIAZEPINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2008-03-27 WO disclosed