SCHEMBL8202847

SCHEMBL8202847

COC(=O)[C@@H]1CCCOc2ccc(cc2)C[C@H](N)C(=O)N[C@@H](C(C)C)C(=O)N1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CAPN2 P17655 4/20 0.46
MMP2 P08253 10/20 0.45
MMP7 P09237 10/20 0.45
MMP3 P08254 10/20 0.45
MMP9 P14780 4/20 0.45
MMP13 P45452 2/20 0.45
MMP12 P39900 1/20 0.45
MMP1 P03956 9/20 0.45
ADAM17 P78536 8/20 0.45
MMP8 P22894 1/20 0.41
MMP14 P50281 1/20 0.41
MMP15 P51511 1/20 0.41
MMP16 P51512 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL931143 0.99 CAPN2 (0.45) CAPN2MMP2MMP7MMP3MMP9
Hydrochloric Acid SCHEMBL931142 0.98 CAPN2 (0.45) CAPN2MMP2MMP7MMP3MMP9
SCHEMBL8205365 0.97 CAPN2 (0.49) CAPN2MMP2MMP7MMP3MMP9
SCHEMBL8203297 0.87 CAPN2 (0.52) CAPN2MMP2MMP7MMP3MMP9
SCHEMBL12943113 0.87 CAPN2 (0.51) CAPN2MMP2MMP7MMP3MMP9
Hydrochloric Acid SCHEMBL929978 0.87 CAPN2 (0.51) CAPN2MMP2MMP7MMP3MMP9
SCHEMBL12943095 0.84 CAPN2 (0.53) CAPN2MMP2MMP7MMP3MMP9
SCHEMBL8206145 0.84 MMP2 (0.44) CAPN2MMP2MMP7MMP3MMP9
SCHEMBL931289 0.83 CAPN2 (0.54) CAPN2MMP2MMP7MMP3MMP9
SCHEMBL15869947 0.83 CAPN2 (0.44) CAPN2MMP2MMP7MMP3MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008048121-A2 MACROCYCLIC CYSTEINE PROTEASE INHIBITORS AND COMPOSITIONS THEREOF LINCOLN UNIVERSITY (NZ) 2008-04-24 WO disclosed