SCHEMBL820394

SCHEMBL820394

Fc1c(F)c(F)c2[nH]ccc2c1F

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CCR8 P51685 1/20 0.37
KMT2A Q03164 1/20 0.36
TNF P01375 1/20 0.35
RIPK1 Q13546 1/20 0.35
P2RX7 Q99572 2/20 0.31
GRIN2D O15399 1/20 0.31
GRIN3B O60391 1/20 0.31
GRIN1 Q05586 1/20 0.31
GRIN2A Q12879 1/20 0.31
GRIN2B Q13224 1/20 0.31
GRIN2C Q14957 1/20 0.31
GRIN3A Q8TCU5 1/20 0.31
KDM4E B2RXH2 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
HSD17B10 Q99714 1/20 0.31
GPR84 Q9NQS5 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27560570 0.97 CCR8 (0.36) CCR8KMT2ATNFRIPK1P2RX7
SCHEMBL18876060 0.81 CCR8 (0.32) CCR8KMT2ATNFRIPK1KDM4E
SCHEMBL2535144 0.73 P2RX7 (0.40) CCR8KMT2ATNFRIPK1P2RX7
SCHEMBL18876042 0.73 TNF (0.36) CCR8KMT2ATNFRIPK1P2RX7
SCHEMBL12219421 0.73 CCR8 (0.50) CCR8KMT2ATNFRIPK1KDM4E
SCHEMBL27269505 0.72
SCHEMBL13991817 0.71 CCR8 (0.36) CCR8KMT2AKDM4ESMN1; SMN2HSD17B10
SCHEMBL28094729 0.70 CFB (0.45) P2RX7
SCHEMBL12748352 0.70 TNF (0.38) CCR8KMT2ATNFRIPK1P2RX7
SCHEMBL27260936 0.69 P2RX7 (0.30) P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 303 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2064248-B1 PREPARATION OF POLYMERIZATION CATALYST ACTIVATORS UTILIZING INDOLE-MODIFIED SILICA SUPPORTS EXXONMOBIL CHEMICAL PATENTS INC (US) 2018-10-10 EP claimed
CN-101511879-B Preparation of polymerization catalyst activators utilizing indole-modified silica supports EXXON MOBIL CHEM PATENTS INC 2012-07-25 CN claimed
CN-1659193-B Polymerization catalyst activators, methods of making, and their use in polymerization processes DOW GLOBAL TECHNOLOGIES INC 2012-06-20 CN claimed
US-7741417-B2 Preparation of polymerization catalyst activators utilizing indole-modified silica supports EXXONMOBIL CHEMICAL PATENTS INC. (US) 2010-06-22 US claimed
CN-101511879-A Preparation of polymerization catalyst activators utilizing indole-modified silica supports EXXONMOBIL CHEM PATENTS INC (US) 2009-08-19 CN claimed
EP-2064248-A1 PREPARATION OF POLYMERIZATION CATALYST ACTIVATORS UTILIZING INDOLE-MODIFIED SILICA SUPPORTS ExxonMobil Chemical Patents Inc. (US) 2009-06-03 EP claimed
WO-2008027116-A1 PREPARATION OF POLYMERIZATION CATALYST ACTIVATORS UTILIZING INDOLE-MODIFIED SILICA SUPPORTS EXXONMOBIL CHEMICAL PATENTS INC. (US) 2008-03-06 WO claimed
US-7220695-B2 Supported activator EXXONMOBIL CHEMICAL PATENTS INC. (US) 2007-05-22 US claimed
US-20070055028-A1 Preparation of polymerization catalyst activators utilizing indole-modified silica supports EXXONMOBIL CHEMICAL PATENTS INC. 2007-03-08 US claimed
US-6989341-B2 Halogen substituted catalyst system for olefin polymerization UNIVATION TECHNOLOGIES, LLC (US) 2006-01-24 US claimed
EP-1517932-A2 HETEROCYCLIC NITROGEN-CONTAINING ACTIVATORS AND CATALYST SYSTEMS FOR OLEFIN POLYMERIZATION Univation Technologies LLC (US) 2005-03-30 EP claimed
EP-1517930-A2 POLYMERIZATION CATALYST ACTIVATORS, METHOD OF PREPARING AND THEIR USE IN POLYMERIZATION PROCESSES Univation Technologies LLC (US) 2005-03-30 EP claimed
EP-1517931-A1 HALOGEN SUBSTITUTED CATALYST SYSTEM FOR OLEFIN POLYMERIZATION Univation Technologies, LLC (US) 2005-03-30 EP claimed
US-6858689-B2 Polymerization catalyst activators, method of preparing, and their use in polymerization processes UNIVATION TECHNOLOGIES, LLC (US) 2005-02-22 US claimed
US-20040167016-A1 Polymerization catalyst activators, method of preparing, and their use in polymerization processes HOLTCAMP MATTHEW W (US) 2004-08-26 US claimed
US-20040127348-A1 Halogen substituted catalyst system for olefin polymerization UNIVATION TECHNOLOGIES, LLC 2004-07-01 US claimed
US-6703338-B2 HETEROCYCLIC COMPOUND COMBINED WITH ALUMOXANE OR ALKYLALUMINUM UNIVATION TECHNOLOGIES, LLC 2004-03-09 US claimed
WO-2004003031-A2 POLYMERIZATION CATALYST ACTIVATORS, METHOD OF PREPARING AND THEIR USE IN POLYMERIZATION PROCESSES UNIVATION TECHNOLOGIES, LLC (US) 2004-01-08 WO claimed
WO-2004003037-A1 HALOGEN SUBSTITUTED CATALYST SYSTEM FOR OLEFIN POLYMERIZATION UNIVATION TECHNOLOGIES, LLC. (US) 2004-01-08 WO claimed
WO-2004003032-A2 HETEROCYCLIC NITROGEN-CONTAINING ACTIVATORS AND CATALYST SYSTEMS FOR OLEFIN POLYMERIZATION UNIVATION TECHNOLOGIES, LLC (US) 2004-01-08 WO claimed