SCHEMBL8204745

SCHEMBL8204745

O=C(/C=C/c1ccc(OCCCBr)cc1)NO

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 9/20 0.58
HDAC3 O15379 7/20 0.58
HDAC1 Q13547 6/20 0.58
HDAC2 Q92769 6/20 0.58
HDAC6 Q9UBN7 6/20 0.58
HDAC4 P56524 4/20 0.55
HDAC7 Q8WUI4 3/20 0.55
HDAC10 Q969S8 3/20 0.55
HDAC11 Q96DB2 3/20 0.55
HDAC9 Q9UKV0 3/20 0.55
HDAC5 Q9UQL6 3/20 0.55
SMN1; SMN2 Q16637 2/20 0.50
RAB9A P51151 1/20 0.50
SAE1 Q9UBE0 1/20 0.50
UBA2 Q9UBT2 1/20 0.50
KMT2A Q03164 2/20 0.49
MEN1 O00255 1/20 0.49
RECQL P46063 1/20 0.49
CYP3A4 P08684 1/20 0.49
NCOR2 Q9Y618 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11278302 0.84 THRB (0.56) KMT2AMEN1
SCHEMBL11278299 0.84 THRB (0.56) KMT2AMEN1
SCHEMBL11023543 0.84 CA12 (0.55) SMN1; SMN2SAE1UBA2KMT2ACYP3A4
SCHEMBL11023539 0.84 CA12 (0.55) SMN1; SMN2SAE1UBA2KMT2ACYP3A4
SCHEMBL29014252 0.80 MAOB (0.71)
SCHEMBL29181747 0.80 MAOB (0.71)
SCHEMBL28928327 0.80 THRB (0.54)
SCHEMBL28669971 0.79 CA12 (0.54) SAE1UBA2CYP3A4
SCHEMBL16774250 0.78 CA12 (0.53) HDAC8HDAC3HDAC1HDAC2HDAC6
SCHEMBL2993109 0.78 NPC1 (0.68) RAB9AKMT2ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008040934-A1 HDAC INHIBITORS CHROMA THERAPEUTICS LTD. (GB) 2008-04-10 WO disclosed