SCHEMBL8205167

SCHEMBL8205167

CNC1=N[C@H](Cc2ccc3ccccc3c2)CO1

nearest known ligand 0.65

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 4/20 0.41
CYP1A2 P05177 1/20 0.39
CYP2A6 P11509 1/20 0.39
NPC1 O15118 1/20 0.36
POLB P06746 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
MAPT P10636 1/20 0.36
CYP2D6 P10635 1/20 0.36
NFKB1 P19838 1/20 0.36
ACHE P22303 1/20 0.36
AIMP2 Q13155 1/20 0.36
HRH3 Q9Y5N1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8195189 0.83 TAAR1 (0.59) TAAR1NPC1POLBRAB9ASMN1; SMN2
SCHEMBL3616587 0.79 TAAR1 (0.68) TAAR1
SCHEMBL3616582 0.79 TAAR1 (0.68) TAAR1
SCHEMBL3619604 0.79 TAAR1 (0.68) TAAR1
SCHEMBL8207545 0.73 SLC6A4 (0.41) TAAR1MAPT
SCHEMBL8210582 0.73 TAAR1 (0.60) TAAR1
SCHEMBL28262128 0.70 CYP1A2 (0.44) TAAR1CYP1A2CYP2A6CYP2D6NFKB1
SCHEMBL19555052 0.69 CYP1A2 (0.40) TAAR1CYP1A2CYP2A6CYP2D6NFKB1
SCHEMBL14498435 0.69 MAPT (0.41) TAAR1NPC1POLBRAB9ASMN1; SMN2
SCHEMBL27838363 0.69 MAPT (0.67) TAAR1NPC1POLBRAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008092785-A1 NOVEL 2-AMINOOXAZOLINES AS TAAR1 LIGANDS FOR CNS DISORDERS F. HOFFMANN-LA ROCHE AG (CH) 2008-08-07 WO disclosed