SCHEMBL28262128

SCHEMBL28262128

C1=NC(Cc2ccc3ccccc3c2)CO1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.44
CYP2A6 P11509 1/20 0.44
SLC6A2 P23975 4/20 0.38
SLC6A4 P31645 4/20 0.38
SLC6A3 Q01959 4/20 0.38
KMT2A Q03164 1/20 0.37
CYP2D6 P10635 1/20 0.37
NFKB1 P19838 1/20 0.37
TAAR1 Q96RJ0 1/20 0.37
ACHE P22303 1/20 0.37
HRH3 Q9Y5N1 1/20 0.36
HTR2A P28223 2/20 0.36
HTR2C P28335 2/20 0.36
HTR2B P41595 2/20 0.36
HTR7 P34969 1/20 0.36
HTR3A P46098 1/20 0.36
HTR4 Q13639 1/20 0.36
KDM1A O60341 1/20 0.35
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21056505 0.82 TAAR1 (0.38) TAAR1HRH3CYP19A1
SCHEMBL21056496 0.81 TAAR1 (0.38) TAAR1
SCHEMBL15823752 0.80 TAAR1 (0.50) TAAR1
SCHEMBL3128078 0.80 TAAR1 (0.50) TAAR1
SCHEMBL21056498 0.76 TAAR1 (0.40) TAAR1
SCHEMBL19555052 0.74 CYP1A2 (0.40) CYP1A2CYP2A6SLC6A2SLC6A4SLC6A3
SCHEMBL845625 0.73 CYP1A2 (0.48) CYP1A2CYP2A6SLC6A2SLC6A4SLC6A3
SCHEMBL31454831 0.73 CYP1A2 (0.48) CYP1A2CYP2A6SLC6A2SLC6A4SLC6A3
SCHEMBL3619604 0.73 TAAR1 (0.68) TAAR1
SCHEMBL3616582 0.73 TAAR1 (0.68) TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109071518-A Oxazoline vacation dimer, medical composition and its use 普渡制药公司 2018-12-21 CN disclosed