SCHEMBL8205302

SCHEMBL8205302

CC(C)(c1cc(N2CCOCC2)nc(-c2ccc(N)cc2)n1)S(=O)(=O)c1ccncc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.48
PIK3CA P42336 6/20 0.48
MTOR P42345 5/20 0.48
PIK3R1 P27986 2/20 0.48
ATR Q13535 5/20 0.45
CYP2C9 P11712 4/20 0.45
CYP2C19 P33261 3/20 0.45
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
CYP1A2 P05177 2/20 0.45
ALDH1A1 P00352 1/20 0.45
MAPT P10636 1/20 0.44
TSHR P16473 1/20 0.44
MAPK1 P28482 1/20 0.44
HSD17B10 Q99714 1/20 0.44
PIK3CB P42338 2/20 0.44
PIK3CG P48736 2/20 0.44
HTT P42858 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.43
CYP3A4 P08684 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8214750 0.89 MTOR (0.50) NPSR1PIK3CAMTORPIK3R1ATR
SCHEMBL3607318 0.86 PIK3CA (0.58) NPSR1PIK3CAMTORPIK3R1ATR
SCHEMBL3601618 0.86 PDCD1 (0.57) PIK3CAMTORATRPIK3CD
SCHEMBL11926804 0.85 PIK3CA (0.51) NPSR1PIK3CAMTORPIK3R1ATR
SCHEMBL8219150 0.81 HRH4 (0.44) NPSR1PIK3CAMTORPIK3R1ATR
SCHEMBL8214586 0.80 NPSR1 (0.47) NPSR1PIK3CAMTORPIK3R1ATR
SCHEMBL3923677 0.77 ATR (0.59) PIK3CAMTORPIK3R1ATRHTT
SCHEMBL740453 0.77 PIK3CA (0.60) PIK3CAMTORATRPIK3CD
SCHEMBL3605539 0.76 PIK3CA (0.56) PIK3CAMTORPIK3R1ATRPIK3CD
SCHEMBL3597950 0.76 PIK3CA (0.56) PIK3CAMTORATRPIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008023159-A1 MORPHOLINO PYRIMIDINE DERIVATIVES USEFUL IN THE TREATMENT OF PROLIFERATIVE DISORDERS ASTRAZENECA AB (SE) 2008-02-28 WO disclosed