SCHEMBL8205632

SCHEMBL8205632

O=C1NC(=O)c2c(CCO)ccc3cccc1c23

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 3/20 0.54
NPSR1 Q6W5P4 2/20 0.41
CDK2 P24941 3/20 0.41
CCNE2 O96020 2/20 0.41
CDK4 P11802 2/20 0.41
CCND1 P24385 2/20 0.41
CCNE1 P24864 2/20 0.41
HEXA P06865 1/20 0.39
HEXB P07686 1/20 0.39
GAA P10253 2/20 0.37
RXFP1 Q9HBX9 1/20 0.37
MEN1 O00255 4/20 0.36
KMT2A Q03164 4/20 0.36
RGS12 O14924 1/20 0.36
USP2 O75604 1/20 0.36
CYP1A2 P05177 1/20 0.36
POLB P06746 1/20 0.36
CYP3A4 P08684 1/20 0.36
MAPT P10636 1/20 0.36
THRB P10828 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8880740 0.90 PARP1 (0.50) PARP1NPSR1CDK2CCNE2CDK4
SCHEMBL11204216 0.88 PARP1 (0.58) PARP1NPSR1CDK2CCNE2CDK4
SCHEMBL11210705 0.87 PARP1 (0.56) PARP1NPSR1CDK2CCNE2CDK4
SCHEMBL19895278 0.85 PARP1 (0.54) PARP1NPSR1GAAMEN1KMT2A
SCHEMBL28257840 0.85 PARP1 (0.54) PARP1NPSR1CDK2HEXAHEXB
Hydrochloric Acid SCHEMBL28259370 0.84 PARP1 (0.53) PARP1NPSR1CDK2HEXAHEXB
SCHEMBL16116423 0.83 PARP1 (0.59) PARP1NPSR1CDK4CCND1GAA
SCHEMBL28174605 0.83 PARP1 (0.51) PARP1NPSR1MEN1KMT2ARGS12
SCHEMBL9556433 0.83 PARP1 (0.51) PARP1NPSR1CDK2CCNE2CDK4
SCHEMBL28287598 0.83 PARP1 (0.51) PARP1NPSR1CDK2HEXAHEXB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6096758-A 3-METHYLIMIDAZOPYRIDINES USED FOR THE TREATMENT OF GASTROINTESTINAL DISORDERS BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 2000-08-01 US disclosed
EP-0359431-A2 Halomethyl-1,3,5-triazines containing a sensitizer moiety MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1990-03-21 EP disclosed