SCHEMBL8880740

SCHEMBL8880740

O=C1NC(=O)c2c(CCCCO)ccc3cccc1c23

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 3/20 0.50
CDK4 P11802 6/20 0.40
CCND1 P24385 6/20 0.40
CCNE2 O96020 5/20 0.40
CCNE1 P24864 5/20 0.40
CDK2 P24941 5/20 0.40
NPSR1 Q6W5P4 2/20 0.38
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
HEXA P06865 1/20 0.36
HEXB P07686 1/20 0.36
GAA P10253 2/20 0.35
RXFP1 Q9HBX9 1/20 0.35
PRKACA P17612 2/20 0.35
PRKACG P22612 2/20 0.35
PRKACB P22694 2/20 0.35
CAMK2B Q13554 2/20 0.35
CAMK2G Q13555 2/20 0.35
CAMK2D Q13557 2/20 0.35
CAMK2A Q9UQM7 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11204216 0.93 PARP1 (0.58) PARP1CDK4CCND1CCNE2CCNE1
SCHEMBL11210705 0.92 PARP1 (0.56) PARP1CDK4CCND1CCNE2CCNE1
SCHEMBL8205632 0.90 PARP1 (0.54) PARP1CDK4CCND1CCNE2CCNE1
SCHEMBL15557200 0.88 PARP1 (0.51) PARP1CDK4CCND1CCNE2CCNE1
SCHEMBL19436979 0.86 PARP1 (0.50) PARP1NPSR1MEN1KMT2AATG4B
SCHEMBL28286146 0.86 PARP1 (0.50) PARP1CDK2NPSR1MEN1KMT2A
SCHEMBL21616783 0.86 PARP1 (0.50) PARP1CDK4CCND1CCNE2CCNE1
SCHEMBL29030849 0.85 PARP1 (0.49) PARP1NPSR1ATG4BTDP1
SCHEMBL9556433 0.85 PARP1 (0.51) PARP1CDK4CCND1CCNE2CCNE1
SCHEMBL28287598 0.85 PARP1 (0.51) PARP1CDK2NPSR1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997046525-A1 5-ALKOXY-TRYPTAMINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS 5-HT1D RECEPTOR AGONISTS ALLELIX BIOPHARMACEUTICALS INC. (CA) 1997-12-11 WO disclosed
US-5654431-A EXHIBIT SELECTIVITY TOWARDS 5-HYDROXYTRYPTAMINE RECEPTORS OF BRAIN CELLS ALLELIX BIOPHARMACEUTICALS INC. (CA) 1997-08-05 US disclosed