SCHEMBL8206271

SCHEMBL8206271

c1coc(COCCCOCCCOCc2ccco2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.47
MAPT P10636 1/20 0.46
GAA P10253 1/20 0.46
CYP2D6 P10635 1/20 0.43
CHRM2 P08172 1/20 0.40
SLC1A3 P43003 1/20 0.39
SLC1A2 P43004 1/20 0.39
SLC1A1 P43005 1/20 0.39
TDP1 Q9NUW8 2/20 0.38
USP2 O75604 2/20 0.38
HPGD P15428 2/20 0.38
CYP3A4 P08684 1/20 0.38
ALOX15 P16050 1/20 0.38
MAPK1 P28482 1/20 0.37
KDM4E B2RXH2 1/20 0.37
LMNA P02545 1/20 0.37
HTT P42858 1/20 0.37
EPHX2 P34913 1/20 0.36
POLB P06746 2/20 0.36
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15087211 0.89 ALDH1A1 (0.52) ALDH1A1MAPTGAACYP2D6CHRM2
SCHEMBL1287680 0.86 ALDH1A1 (0.47) ALDH1A1MAPTGAACYP2D6USP2
SCHEMBL8905002 0.86 ALDH1A1 (0.47) ALDH1A1MAPTGAACYP2D6CHRM2
SCHEMBL686820 0.86 ALDH1A1 (0.47) ALDH1A1MAPTGAACYP2D6CHRM2
SCHEMBL14230617 0.86 ALDH1A1 (0.43) ALDH1A1MAPTGAACYP2D6CHRM2
SCHEMBL10934229 0.85 MAPT (0.42) ALDH1A1MAPTGAACYP2D6CHRM2
SCHEMBL4613994 0.85 ALDH1A1 (0.46) ALDH1A1MAPTGAACYP2D6USP2
SCHEMBL29260920 0.85 ALDH1A1 (0.46) ALDH1A1MAPTGAACYP2D6CHRM2
SCHEMBL8906026 0.85 ALDH1A1 (0.46) ALDH1A1MAPTGAACYP2D6CHRM2
SCHEMBL891457 0.84 ALDH1A1 (0.55) ALDH1A1MAPTGAACYP2D6CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019073431-A1 AN IMPROVED PROCESS FOR THE PREPARATION OF APREMILAST AND ITS INTERMEDIATE Piramal Enterprises Limited (IN) 2019-04-18 WO claimed
WO-2019073431-A1 AN IMPROVED PROCESS FOR THE PREPARATION OF APREMILAST AND ITS INTERMEDIATE Piramal Enterprises Limited (IN) 2019-04-18 WO disclosed
US-6130195-A TETRAHYDROFURFURYL ALCOHOL AND 3-METHOXY-3-METHYL BUTANOL. KYZEN CORPORATION (US) 2000-10-10 US disclosed