SCHEMBL8206428

SCHEMBL8206428

Nc1sc2c(c1C(=O)NCc1ccc3c(c1)OCO3)CCCC2

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.58
CRHBP P24387 1/20 0.58
RECQL P46063 1/20 0.58
CRHR2 Q13324 1/20 0.58
ALDH2 P05091 1/20 0.56
TAAR1 Q96RJ0 2/20 0.55
ALDH1A1 P00352 6/20 0.54
MEN1 O00255 5/20 0.54
KMT2A Q03164 5/20 0.54
KDM4E B2RXH2 4/20 0.54
HPGD P15428 4/20 0.54
MAPT P10636 4/20 0.54
HSD17B10 Q99714 4/20 0.54
ALOX15 P16050 3/20 0.54
TSHR P16473 2/20 0.54
POLB P06746 2/20 0.54
SMN1; SMN2 Q16637 2/20 0.54
USP2 O75604 1/20 0.54
GAA P10253 1/20 0.54
CASP1 P29466 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7421905 0.82 ALDH1A1 (0.55) ALDH1A1MEN1KMT2AKDM4EHPGD
SCHEMBL7426573 0.82 KDM4E (0.61) TP53RECQLALDH2ALDH1A1MEN1
SCHEMBL8207916 0.80 TAAR1 (0.78) TAAR1ALDH1A1MEN1KMT2AKDM4E
SCHEMBL7889391 0.80 KMT2A (0.68) TP53ALDH1A1MEN1KMT2AKDM4E
SCHEMBL14829398 0.79 TAAR1 (0.76) TAAR1ALDH1A1MEN1KMT2AKDM4E
SCHEMBL20915168 0.79 MAPT (0.64) TP53TAAR1ALDH1A1MEN1KMT2A
SCHEMBL135251 0.79 FLT3 (0.62) RECQLALDH1A1MEN1KMT2AKDM4E
SCHEMBL8206811 0.79 TAAR1 (0.62) RECQLTAAR1ALDH1A1MEN1KMT2A
SCHEMBL8210444 0.79 KMT2A (0.61) TP53RECQLTAAR1ALDH1A1MEN1
Bicarbonate SCHEMBL7421513 0.78 ALDH1A1 (0.56) TP53CRHBPRECQLCRHR2ALDH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6143777-A ENZYME INHIBITORS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-07 US disclosed