SCHEMBL8208044

SCHEMBL8208044

CCC[C@@H]1NC(=O)[C@@H](NS(=O)(=O)c2ccc(F)cc2)Cc2ccc(cc2)OCCCC[C@@H](CO)NC1=O

nearest known ligand 0.59

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CAPN2 P17655 11/20 0.59
CPB2 Q96IY4 2/20 0.39
MMP1 P03956 3/20 0.36
MMP2 P08253 3/20 0.36
MMP3 P08254 3/20 0.36
MMP7 P09237 3/20 0.36
F2 P00734 1/20 0.35
F10 P00742 1/20 0.35
PLG P00747 1/20 0.35
KLKB1 P03952 1/20 0.35
PROC P04070 1/20 0.35
ADAM17 P78536 2/20 0.35
PSMB8 P28062 1/20 0.34
PSMB5 P28074 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL931525 0.90 CAPN2 (0.63) CAPN2MMP1MMP2MMP3MMP7
SCHEMBL8202837 0.88 CAPN2 (0.75) CAPN2CPB2MMP1MMP2MMP3
SCHEMBL8206129 0.78 CAPN2 (0.79) CAPN2CPB2MMP1MMP2MMP3
SCHEMBL931065 0.77 CAPN2 (0.58) CAPN2MMP1MMP2MMP3MMP7
SCHEMBL8202872 0.75 CAPN2 (0.75) CAPN2CPB2MMP1MMP2MMP3
SCHEMBL930611 0.75 CAPN2 (1.00) CAPN2CPB2MMP1MMP2MMP3
SCHEMBL8208872 0.75 CAPN2 (1.00) CAPN2CPB2MMP1MMP2MMP3
SCHEMBL8208871 0.74 CAPN2 (0.74) CAPN2CPB2MMP1MMP2MMP3
SCHEMBL931644 0.72 CAPN2 (1.00) CAPN2CPB2MMP1MMP2MMP3
SCHEMBL930019 0.72 CAPN2 (0.74) CAPN2CPB2MMP1MMP2MMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008048121-A2 MACROCYCLIC CYSTEINE PROTEASE INHIBITORS AND COMPOSITIONS THEREOF LINCOLN UNIVERSITY (NZ) 2008-04-24 WO disclosed