SCHEMBL8208743

SCHEMBL8208743

Nc1nc2nc(Cc3ccc(-c4ccccc4)s3)[nH]c2c(=O)[nH]1

nearest known ligand 0.64

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PNP P00491 10/20 0.64
FGFR1 P11362 1/20 0.54
FGFR2 P21802 1/20 0.54
CYP2E1 P05181 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2A6 P11509 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2B6 P20813 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9434519 0.81 PNP (0.64) PNPFGFR1FGFR2
SCHEMBL3300185 0.81 PNP (0.64) PNPFGFR1FGFR2
SCHEMBL4963414 0.81 PNP (0.64) PNPFGFR1FGFR2
SCHEMBL18248 0.79 PNP (1.00) PNPFGFR1FGFR2
SCHEMBL4966173 0.78 PNP (0.63) PNPFGFR1FGFR2CYP2A6
SCHEMBL4962855 0.77 PNP (1.00) PNPFGFR1FGFR2
Hydrochloric Acid SCHEMBL17186372 0.76 PNP (0.97) PNPFGFR1FGFR2
SCHEMBL9960811 0.75 PNP (0.71) PNPFGFR1FGFR2
SCHEMBL1938287 0.74 PNP (0.71) PNPFGFR1FGFR2
SCHEMBL9283418 0.73 PNP (0.66) PNPFGFR1FGFR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6096724-A O(6)-ALKYLGUANINE-DNA ALKYLTRANSFERASE (ATASE) ENZYME INHIBITORS CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 2000-08-01 US disclosed