SCHEMBL8209101

SCHEMBL8209101

CC(C)C[C@@H]1NC(=O)[C@@H](NC(=O)OC(C)(C)C)Cc2ccc(cc2)OC/C=C/COC[C@@H](C(=O)O)NC1=O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CAPN2 P17655 9/20 0.49
TMPRSS2 O15393 4/20 0.43
F2 P00734 4/20 0.43
HPN P05981 4/20 0.43
ST14 Q9Y5Y6 4/20 0.43
HGFAC Q04756 2/20 0.43
CTSD P07339 2/20 0.43
BACE1 P56817 2/20 0.43
PSMB11 A5LHX3 2/20 0.41
PSMA7 O14818 2/20 0.41
PSMB1 P20618 2/20 0.41
PSMA1 P25786 2/20 0.41
PSMA2 P25787 2/20 0.41
PSMA3 P25788 2/20 0.41
PSMA4 P25789 2/20 0.41
PSMB8 P28062 2/20 0.41
PSMB9 P28065 2/20 0.41
PSMA5 P28066 2/20 0.41
PSMB4 P28070 2/20 0.41
PSMB6 P28072 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12943167 0.93 CAPN2 (0.47) CAPN2TMPRSS2F2HPNST14
SCHEMBL8209212 0.87 CAPN2 (0.48) CAPN2TMPRSS2F2HPNST14
SCHEMBL12943280 0.87 CAPN2 (0.48) CAPN2TMPRSS2F2HPNST14
SCHEMBL17884328 0.85 CAPN2 (0.49) CAPN2TMPRSS2F2HPNST14
SCHEMBL12943281 0.83 CAPN2 (0.49) CAPN2TMPRSS2F2HPNST14
SCHEMBL931569 0.82 CAPN2 (0.55) CAPN2TMPRSS2F2HPNST14
SCHEMBL17884315 0.81 CTSD (0.49) CAPN2CTSDBACE1
SCHEMBL929429 0.79 CAPN2 (0.60) CAPN2TMPRSS2F2HPNST14
SCHEMBL12943118 0.79 CAPN2 (0.51) CAPN2TMPRSS2F2HPNST14
SCHEMBL17884332 0.79 CAPN2 (0.51) CAPN2TMPRSS2F2HPNST14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008048121-A2 MACROCYCLIC CYSTEINE PROTEASE INHIBITORS AND COMPOSITIONS THEREOF LINCOLN UNIVERSITY (NZ) 2008-04-24 WO disclosed