SCHEMBL8209215

SCHEMBL8209215

Cc1ccc(-n2nccn2)c(C(=O)N2CCCN(C(=O)OC(C)(C)C)CC2)c1

nearest known ligand 0.59

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 14/20 0.59
HCRTR1 O43613 12/20 0.59
LMNA P02545 2/20 0.49
MAPT P10636 1/20 0.49
POLB P06746 1/20 0.49
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13208901 0.85 POLB (0.58) HCRTR2HCRTR1LMNAMAPTPOLB
SCHEMBL13789995 0.85 HCRTR1 (0.51) HCRTR2HCRTR1
SCHEMBL2905303 0.85 HCRTR1 (0.51) HCRTR2HCRTR1
SCHEMBL2904616 0.85 HCRTR1 (0.51) HCRTR2HCRTR1
SCHEMBL17501812 0.85 HCRTR2 (0.65) HCRTR2HCRTR1
SCHEMBL19894076 0.85 HCRTR2 (0.48) HCRTR2HCRTR1LMNAMAPT
SCHEMBL17539230 0.84 HCRTR2 (0.56) HCRTR2HCRTR1
SCHEMBL17539260 0.84 HCRTR2 (0.56) HCRTR2HCRTR1
SCHEMBL2358754 0.84 HCRTR2 (0.64) HCRTR2HCRTR1
SCHEMBL17539262 0.84 HCRTR2 (0.64) HCRTR2HCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016020403-A1 PREPARATION OF A BENZOIC ACID DERIVATIVE AND ITS USE FOR THE PREPARATION OF SUVOREXANT SANDOZ AG (CH) 2016-02-11 WO disclosed
WO-2016020403-A1 PREPARATION OF A BENZOIC ACID DERIVATIVE AND ITS USE FOR THE PREPARATION OF SUVOREXANT SANDOZ AG (CH) 2016-02-11 WO disclosed
WO-2008008518-A1 SUBSTITUTED DIAZEPAN OREXIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2008-01-17 WO disclosed