SCHEMBL8209422

SCHEMBL8209422

CCCN(C)Cc1ccc(C(=O)NN(c2nc(N)ncc2Cl)C2CCCC2)cc1

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.37
DRD3 P35462 2/20 0.37
TRPV1 Q8NER1 1/20 0.37
F10 P00742 6/20 0.36
TMEM97 Q5BJF2 5/20 0.35
SIGMAR1 Q99720 5/20 0.35
ACVR1 Q04771 2/20 0.35
LCK P06239 1/20 0.35
JAK3 P52333 1/20 0.35
HIF1A Q16665 1/20 0.33
EPAS1 Q99814 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
THRB P10828 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8206710 0.95 TMEM97 (0.39) DRD2DRD3TRPV1F10TMEM97
SCHEMBL8206008 0.93 TMEM97 (0.38) DRD2DRD3TRPV1F10TMEM97
SCHEMBL8206010 0.93 F10 (0.42) DRD2DRD3F10TMEM97SIGMAR1
SCHEMBL8205988 0.90 ACVR1 (0.43) F10ACVR1LCKJAK3
SCHEMBL8205845 0.90 HDAC1 (0.41) DRD2DRD3TMEM97SIGMAR1
SCHEMBL8209425 0.89 S1PR1 (0.35) DRD2DRD3F10ACVR1LCK
SCHEMBL8203780 0.88 SIGMAR1 (0.44) DRD2DRD3TMEM97SIGMAR1
SCHEMBL8193280 0.88 HDAC6 (0.42) F10ACVR1LCKJAK3
SCHEMBL8193482 0.88 ITK (0.41) TRPV1ACVR1LCKJAK3
SCHEMBL8198832 0.87 HDAC6 (0.43) DRD2DRD3ACVR1LCKJAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008052934-A1 NOVEL SUBSTITUTED PYRIMIDINES AS CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2008-05-08 WO disclosed