SCHEMBL8209613

SCHEMBL8209613

CO[C@@H]1CNC[C@H]1Cc1csc(NC(=O)OC(C)(C)C)n1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SIRT1 Q96EB6 1/20 0.47
PI4KB Q9UBF8 1/20 0.38
SMN1; SMN2 Q16637 4/20 0.36
KMT2A Q03164 2/20 0.35
CCR2 P41597 4/20 0.35
TSHR P16473 1/20 0.35
MAPK1 P28482 1/20 0.35
HDAC3 O15379 2/20 0.34
HDAC1 Q13547 2/20 0.34
HDAC2 Q92769 2/20 0.34
HDAC10 Q969S8 2/20 0.34
HDAC8 Q9BY41 2/20 0.34
LMNA P02545 2/20 0.33
KCNH2 Q12809 1/20 0.33
LCK P06239 1/20 0.33
ALDH1A1 P00352 1/20 0.33
ABCB1 P08183 1/20 0.33
MEN1 O00255 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2600855 0.87 SIRT1 (0.46) SIRT1PI4KBSMN1; SMN2KMT2ACCR2
SCHEMBL2600851 0.87 SIRT1 (0.46) SIRT1PI4KBSMN1; SMN2KMT2ACCR2
SCHEMBL9071272 0.76 SIRT1 (0.49) SIRT1PI4KBSMN1; SMN2KMT2ACCR2
SCHEMBL2600845 0.75 SIRT1 (0.49) SIRT1PI4KBSMN1; SMN2KMT2ACCR2
SCHEMBL1742461 0.75 PTPRB (0.49) SIRT1PI4KBSMN1; SMN2KMT2ACCR2
SCHEMBL2175797 0.74 SMN1; SMN2 (0.50) SIRT1PI4KBSMN1; SMN2KMT2ACCR2
SCHEMBL1030124 0.74 PI4KB (0.50) SIRT1PI4KBSMN1; SMN2KMT2ACCR2
SCHEMBL2600847 0.74 SIRT1 (0.46) SIRT1PI4KBSMN1; SMN2KMT2ACCR2
SCHEMBL2600849 0.74 SIRT1 (0.46) SIRT1PI4KBSMN1; SMN2KMT2ACCR2
SCHEMBL7419507 0.74 SMN1; SMN2 (0.56) SIRT1SMN1; SMN2KMT2ATSHRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008042353-A1 POTENT AND HIGHLY SELECTIVE HETEROAROMATIC INHIBITORS OF NEURONAL NITRIC OXIDE SYNTHASE NORTHWESTERN UNIVERSITY (US) 2008-04-10 WO disclosed