SCHEMBL8211530

SCHEMBL8211530

CCCCOC(=O)c1c(N)cccc1Br

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.60
HSD17B10 Q99714 2/20 0.60
KDM4E B2RXH2 1/20 0.54
POLB P06746 1/20 0.54
TSHR P16473 6/20 0.51
L3MBTL1 Q9Y468 3/20 0.51
TDP1 Q9NUW8 2/20 0.51
LMNA P02545 3/20 0.51
CYP3A4 P08684 3/20 0.51
CYP1A2 P05177 2/20 0.51
CYP2C19 P33261 2/20 0.51
CYP2C9 P11712 1/20 0.51
PDE4D Q08499 1/20 0.51
ESR1 P03372 4/20 0.49
MAPK1 P28482 3/20 0.46
TP53 P04637 1/20 0.46
NPC1 O15118 1/20 0.46
MAPT P10636 1/20 0.46
RAB9A P51151 1/20 0.46
CYP2D6 P10635 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3860479 0.89 ALDH1A1 (0.69) ALDH1A1HSD17B10KDM4EPOLBTSHR
SCHEMBL1189107 0.84 CA12 (0.56) ALDH1A1HSD17B10KDM4EPOLBTSHR
SCHEMBL30327304 0.84 TSHR (0.66) ALDH1A1HSD17B10KDM4EPOLBTSHR
SCHEMBL4628037 0.84 TSHR (0.66) ALDH1A1HSD17B10KDM4EPOLBTSHR
SCHEMBL8894641 0.84 ALDH1A1 (0.75) ALDH1A1HSD17B10KDM4EPOLBTSHR
SCHEMBL30755640 0.84 TSHR (0.53) ALDH1A1HSD17B10TSHRL3MBTL1TDP1
SCHEMBL8804913 0.82 ALDH1A1 (0.60) ALDH1A1HSD17B10KDM4EPOLBTSHR
SCHEMBL17493148 0.82 ALDH1A1 (0.60) ALDH1A1HSD17B10KDM4EPOLBTSHR
SCHEMBL8007082 0.81 ALDH1A1 (0.67) ALDH1A1HSD17B10KDM4EPOLBTSHR
SCHEMBL4627373 0.80 TSHR (0.60) ALDH1A1HSD17B10KDM4EPOLBTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0979227-A1 4,1-BENZOXAZEPINES, THEIR ANALOGUES, AND THEIR USE AS SOMATOSTATIN AGONISTS Takeda Chemical Industries, Ltd. (JP) 2000-02-16 EP disclosed
WO-1998047882-A1 4,1-BENZOXAZEPINES, THEIR ANALOGUES, AND THEIR USE AS SOMATOSTATIN AGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-10-29 WO disclosed