SCHEMBL8212290

SCHEMBL8212290

C[N+](C)(C)Cc1n[nH]c2ccccc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.47
GAA P10253 2/20 0.47
PDPK1 O15530 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP1A2 P05177 1/20 0.44
IDO1 P14902 3/20 0.44
ALDH1A1 P00352 2/20 0.44
ALPL P05186 1/20 0.44
HPGD P15428 1/20 0.44
TTK P33981 1/20 0.44
MAPK10 P53779 1/20 0.44
YTHDC1 Q96MU7 1/20 0.40
STAT3 P40763 1/20 0.40
HIF1A Q16665 1/20 0.40
TRPA1 O75762 1/20 0.39
LRRK2 Q5S007 2/20 0.39
NPC1 O15118 1/20 0.39
TP53 P04637 1/20 0.39
RAB9A P51151 1/20 0.39
FLT3 P36888 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Iodide SCHEMBL1595770 0.98 KDM4E (0.46) KDM4EGAAPDPK1CYP3A4CYP1A2
SCHEMBL254885 0.79 KDM4E (0.52) KDM4EGAAPDPK1CYP3A4CYP1A2
SCHEMBL8206970 0.76 MAP2K4 (0.47)
SCHEMBL3347649 0.76 KDM4E (0.48) KDM4EGAAPDPK1CYP3A4CYP1A2
SCHEMBL12776223 0.76 KDM4E (0.48) KDM4EGAAPDPK1CYP3A4CYP1A2
SCHEMBL730574 0.75 KDM4E (0.52) KDM4EGAAPDPK1CYP3A4CYP1A2
SCHEMBL3061437 0.75 KDM4E (0.52) KDM4EGAAPDPK1CYP3A4CYP1A2
SCHEMBL702375 0.75 PRMT5 (0.61) KDM4EGAAPDPK1CYP3A4CYP1A2
SCHEMBL2227955 0.75 KDM4E (0.52) KDM4EGAAPDPK1CYP3A4CYP1A2
SCHEMBL16182225 0.75 KDM4E (0.52) KDM4EGAAPDPK1CYP3A4CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008040995-A9 INDAZOLES FOR USE AS DPP-IV INHIBITORS PEAKDALE MOLECULAR LTD (GB) 2008-12-31 WO disclosed
WO-2008040995-A1 INDAZOLES FOR USE AS DPP-IV INHIBITORS PEAKDALE MOLECULAR LIMITED (GB) 2008-04-10 WO disclosed