SCHEMBL8213178

SCHEMBL8213178

CC(=O)N1CCC2(CC1)C(=O)N(CC(C)C)C2c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 7/20 0.48
CYP2D6 P10635 3/20 0.42
CYP3A4 P08684 2/20 0.41
ALDH1A1 P00352 2/20 0.41
CYP2C9 P11712 1/20 0.41
TSHR P16473 1/20 0.41
USP2 O75604 1/20 0.41
MAPK1 P28482 1/20 0.40
CYP2C19 P33261 1/20 0.40
CACNA1H O95180 2/20 0.40
GAA P10253 1/20 0.39
GFER P55789 1/20 0.39
OPRK1 P41145 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8218924 0.85 HDAC1 (0.47) TRPV1CYP2D6CYP3A4TSHRUSP2
SCHEMBL8227883 0.75 CACNA1H (0.47) ALDH1A1MAPK1CACNA1H
SCHEMBL8213185 0.72 CACNA1H (0.41) CACNA1H
SCHEMBL26822130 0.71 MDM2 (0.42) CACNA1HOPRK1
SCHEMBL8212405 0.70 CACNA1H (0.71) TRPV1CACNA1H
SCHEMBL12876984 0.70 CACNA1H (0.71) TRPV1CACNA1H
SCHEMBL17888237 0.69 HDAC1 (0.54) MAPK1
SCHEMBL8224879 0.68 HDAC1 (0.44) TRPV1TSHROPRK1
SCHEMBL8208288 0.68 HDAC1 (0.47) TRPV1TSHR
SCHEMBL8227850 0.68 HDAC1 (0.45) TRPV1TSHROPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008033465-A1 AZETIDINONE DERIVATIVES AND METHODS OF USE THEREOF SCHERING CORPORATION (US) 2008-03-20 WO disclosed